Ahụ ike, Preparations
Ntụziaka ndị zuru ezu "Futsisa": egosi maka ojiji, analogs na reviews
Yana ọgwụ nje elekọta mmadụ, antifungal mmadụ n'ụzọ dị irè-enyere ndị ọrịa tufuo ọrịa nke na-kpatara microorganisms susceptible ka ha nọ n'ọrụ umi.
Ugbu a, e nwere ndị a na nnukwu ọnụ ọgụgụ nke ndị dị otú ọgwụ. Ha pharmacological e ji mara mgbe idako. Ma, ọtụtụ ndị ọkachamara nye iwu ndị dị otú ahụ a ọgwụ na ha na-agwọ dị ka "Futsis". Ntuziaka maka ojiji na atụmatụ nke ngwá ọrụ ga-adade ke ihe ndị a n'isiokwu a.
The mejupụtara, na udi ma na nkwakọ
Ọgwụ "Futsis" ntụziaka nke na-agbakwunyere na a ikpo nke katọn, nwere ike zụrụ n'ụdị mbadamba. Ha n'ọrụ mgwa eme dị ka fluconazole. Ọzọkwa na agwọ ọrịa na-agụnye inyeaka mmiri.
E lee ya anya ngwaahịa emepụta doses nke 50, 150, 100 na 200 mg. Mbadamba ke ichekwa 4 iberibe, juru n'ọnụ katọn na ọnya mkpọ, karị.
Na ihe ndị ọzọ ụdị nwere ike zụrụ "Futsis"? Ntuziaka maka ojiji (mbadamba - nke a abụghị naanị ụdị kwuru mmadụ) na-akọ na ndị agwọ ọrịa na-arụpụtara n'ụdị ihe ngwọta maka infusion. The mejupụtara agụnye mbadamba fluconazole na ndị ọzọ Efrata ndị dị otú dị ka microcrystalline cellulose, povidone K30, lactose, talc, magnesium stearate, sodium croscarmellose, sodium starch glycolate na ndị ọzọ.
The ngwọta maka igba ogwu n'akwara injections ahịa na karama nke 100 ml.
Ma ihe ndị jel "Futsis", mgbe ahụ, ọ nwere ike zụta na akpa nke 30 g
Pharmacology agwọ ọrịa
Olee ihe ndị na pụta ụwa ọgwụ "Futsis"? Ngwa ntụziaka na-enye na kwuru pụtara na onye ọ bụla ụdị nwere a akpọ antifungal ọrụ.
Fluconazole bụ a sịntetik emepụta na bụ otu nke thiazole ogige. Nke a ihe onwunwe na-enyere kpochapụ enzymatic ọrụ nke kpọmkwem mmiri nke na-na fungal mkpụrụ ndụ.
Mgbe ọgwụ ọjọọ na-ewute ndu njikọ nke sterol ogige ma nwekwara gbochie na usoro nke na n'ịtụgharị lanosterol ergosterol. Mgbanwe ndị dị otú na cell membranes akwalite cessation nke mmeputakwa nke dịkwa ka usoro ha.
Njirimara nke ọgwụ
Gịnị Njirimara nke ọgwụ ọjọọ, "Futsis"? Ntuziaka maka ojiji (mbadamba nwere otu pharmacological e ji mara dị ka ihe ngwọta na jel) na-ekwu na a agwọ ọrịa e ji mara ala toxicity. Na nke a, na o nweghị ezighị ezi mmetụta na ahụ mmadụ, dị ka nke ọma dị ka a dị ịrịba ama mmetụta na ego nke cytochromes na androgenic homonụ na ọbara plasma.
Pharmacokinetics nke ọgwụ
Ntuziaka "Futsisa" na-ekwu na mgbe na-ewere ọgwụ n'ime ha, ha bụ ndị mara mma ngwa ngwa na-ọma etinye obi gị dum na eriri afọ tract. Dị ka ọkachamara, fluconazole nwere nnukwu bioavailability. Jiri nke nri nwere enweghị mmetụta na absorption usoro nke ngwá ọrụ.
The kacha ịta nke nọ n'ọrụ umi ke ọbara plasma a hụrụ mgbe banyere 60-90 nkeji mgbe ochichi.
E lee ya anya ọgwụ nnọọ nke ọma n'ime ihe ndị mejupụtara nke mmiri ahụ na anụ ahụ. Fluconazole nwekwara-agabiga ọbara-ụbụrụ mgbochi na-etinye uche na cerebrospinal ọmụmụ.
Excretion nke ọgwụ si ọrịa ahụ a rụrụ na mmamịrị. Ya ọkara ndụ bụ banyere 30 awa.
Gịnị kinetic kwa nwere ihe ngwọta "Futsis"? Guide na-ekwu na pharmacokinetics nke ọgwụ mgbe ndinọ intravenously bụ nnọọ iche onu ochichi.
Banyere antifungal mmadụ n'ụdị jel, o nwere otu e ji mara na ọrụ. Karịsịa irè jel-egosipụta onwe ya mgbe dermatophytes na yeasts.
Mgbe Nde ngwa nke ngwá ọrụ, obere nke nọ n'ọrụ gị n'ụlọnga abatakwa n'ọbara. Na nke a, ya kpam kpam eliminates systemic edinam.
Ọkachamara na-a hụrụ na jel anaghị njọ imetụta akpụkpọ ọnọdụ.
egosi
Ntuziaka "Futsisa" na-akọ na ọgwụ a na-eji na ọgwụgwọ nke na-efe efe nke dị iche iche orunótu, nke e mere site microorganisms, igosipụta a elu uche na fluconazole. Dị ka a na-achị, na-ewere ọgwụ họpụtara gynecologists, dermatologists na mycologists.
Ya mere, mgbe na-eji ọgwụ ọjọọ, "Futsis" (mbadamba)? Guide na-akọ na ndị ọgwụ kenyere a:
- mycosis ọrịa, mere na ụkwụ na na ukwu ebe, onychomycosis, tinea na tinea versicolor;
- na-efe efe nke mucous membranes, nke e mere site na fungi nke genus Candida;
- candidal na-efe efe nke dị iche iche ebe (e.g., candidemia, akwadebe candidiasis, na ụdị ndị ọzọ candiduria generalized candidiasis na e mere site ero Candida);
- noninvasive bronchopulmonary candidal na-efe efe;
- ọgwụgwọ nke ala ala na nnukwu iche nke mmamiri candidiasis (ntighari);
- adịghị ala ala candidiasis nke onu mucosa, nke jikọtara yi eze;
- ọgwụgwọ nke histoplasmosis, sporotrichosis na ndị ọzọ na-enwekarị n'ebe ụfọdụ mycoses.
Gịnị ka ebumnuche nke ọnụ na nkwadebe "Futsis" (mbadamba) nwere ike na-kenyere? Ntụziaka na-ekwu na ọgwụ a na-eji maka mgbochi nke nlọghachite na ọrịa na:
- candidal balanitis;
- mmamiri-adịghị ala ala candidiasis;
- cryptococcal na-efe efe nke dị iche iche orunótu;
- fungal-efe efe nke dị iche iche orunótu, ma ọ bụrụ na onye ọrịa na-ata ahụhụ site na immunodeficiency ma ọ bụ na-anata cytostatic na ụzarị ọkụ na ọgwụ.
Ma ihe ngwọta maka infusion ochichi, ntụziaka "Futsisa" na-egosi na nke a ụdị nke ọgwụ na-eji na ọgwụgwọ nke:
- cryptococcal meningitis;
- systemic fungal-efe efe (candidemia, candidal anya na-efe efe candiduria endocardium);
- cryptococcal na-efe efe nke anụ ahụ na akụkụ okuku ume na usoro.
The ọgwụ maka mpụga na ngwa nwere ike na-kenyere mgbe:
- ringworm na-eme ka yist;
- tinea (jock oko,-eme egwuregwu ụkwụ, trichophytosis, pityriasis versicolor na kandidnyh na-efe efe).
contraindications
Gịnị bụ ọgwụgwọ Usoro "Futsis" ọgwụ maka ụmụaka? Guide na-ekwu na ọ bụ ụzọ na okenye na ụmụaka adịghị atụ aro maka ojiji na enwekwukwa uche na onye ọcha nke ọgwụ. Ọzọkwa, ọ bụ na-eji na ọnụnọ nke asọ azole ogige ezigbo na Ọdịdị na fluconazole.
Afọ ole kwesịrị inweta "Futsis Dt" maka ụmụaka? Ntuziaka na-agwa na ot mbadamba na-nnọọ contraindicated maka ọgwụgwọ nke ụmụ ruo 7 afọ, na chụgara - ruo afọ 3.
Ọzọkwa anya ọgwụ a machibidoro iwu na-enweta n'oge ime na ara. Ọ na-adịghị mee ihe maka ọgwụgwọ nke ndị mmadụ na-anata ọgwụgwọ "cisapride" na "terfenadine" na ndị na onye na-arụ ọrụ na-metụtara moto akara na nwere ize ndụ ígwè.
Drug "Futsis Dt": ntuziaka maka ojiji
The agwọ ọrịa na mbadamba ụdị, nakwa dị ka ihe ngwọta na jel ga-eji dị iche iche.
Olee na-ọgwụ ọjọọ, "Futsis 50"? Manual na-ekwu na a ọgwụ na ifịk umi ọdịnaya 50-200 mg a na-eji na-emeso bụghị naanị ndị okenye, ma na-eto eto na-arịa ọrịa nke 3-7 afọ.
Mbadamba na-e mgbe ọ bụla nke ụbọchị ọnụ. The kwa onunu ogwu nke ọgwụ na-zubere maka otu oge na e debere naanị site a dibịa (dabere n'elu ọrịa).
Olee otú iji chụgara mbadamba "Futsis" (50 mg)? Guide na-akọ na tupu ewere a ọgwụ ọ ga-etisasịwo ke nkịtị mmiri (banyere 5 ml).
Ndị na-enwe Genital candidiasis, ọgwụ ozugbo ndinọ na mbadamba nkume nke 150 mg. Iji gbochie a nlọghachite nke mmamiri candidiasis-adịghị ala ala uwa (thrush) ọgwụ na-eji na otu dose, ma naanị otu ugboro a ọnwa.
N'ozuzu, na onunu ogwu n'aka na-adịghị na-ewere dabere na usoro nke ya ngwa, na a na-adịghị agbanwe agbanwe n'oge Transition si parenteral ochichi na onu.
Dosing infusion ngwọta
The ntụziaka "Futsisa" na-akọ na na nkwadebe maka igba ogwu n'akwara ọgwụ nwere 200 mg nke fluconazole na 100 ml nke sodium chloride ngwọta (isotonic).
Tupu iwebata agwọ ọrịa ka ọrịa kwesịrị mmachi oriri nke mmiri na sodium. Ọ na-achọrọ iji tụlee ọdịnaya nke chloride na sodium ion na ngwọta.
N'agbanyeghị enweghị oké ọgwụ incompatibility nke ego na-ekwesịghị weere na ndị ọzọ ọgwụ ọjọọ eme ihe maka infusion.
The ojiji nke jel
Jel "Futsis" nakwa dị ka mbadamba, ọ dị mkpa iji otu ugboro n'ụbọchị. The mpụga gị n'ụlọnga nwayọọ ụlọ akwụkwọ ji agwụ n'ime metụtara akpụkpọ ebe, nakwa dị ka na mpaghara dị gburugburu ha.
Ndị ọkachamara na-na-akọ na iji nweta a ọgwụgwọ mmetụta onye ọrịa na-achọ naanị a obere ego nke jel. Ya nke ọma ụlọ akwụkwọ ji agwụ gafee fungi nke emetụtara n'elu ebe, iji gbochie maceration.
Ugbu a ị maara otú e si eji jel ngwọta na "Futsis" Mbadamba (150 mg). Ntụziaka na-ekwu na usoro onunu ogwu na oge nke ojiji nke onye ọ bụla nke osụk forms kwesịrị ikpebisi ike naanị site ịga dibịa.
mmetụta
Gịnị mmetụta nwere ike ime ka ngwa nke ihe infusion ngwọta, jel na "Futsis 150" mbadamba? Ntụziaka na-ekwu na na ndabere nke ihe ndị a ego, onye ọrịa nwere ike ịzụlite na-esonụ oghom Jeremaya mere:
- inwe isi ọwụwa, mara jijiji, dizziness na ụfụ;
- arrhythmia na tachycardia;
- ọgbụgbọ, abdominal mgbu, vomiting, afọ mgbu, afọ ọsịsa, na ndị ọzọ na;
- Nfụkasị Jeremaya na akpụkpọ n'ụdị alopecia, nsí epidermal necrosis, itching, anụ ọkụ ọkụ, aṅụ, edema, Stevens-Johnson syndrome.
Ọzọkwa, na ojiji nke a ọgwụ ike imetụta arụmọrụ nke laabu ule (neutropenia, leukopenia, agranulocytosis, hypokalemia, thrombocytopenia, triglycerides na cholesterol n'ime ọbara).
Ndị a mmetụta achọ ozugbo cessation nke "Futsisa".
ikpe nke ovadozu
Bụrụ na nke ovadozu ma ọ bụ ihe ngwọta "Futsis" mkpụrụ ọgwụ a ndidi nwere ike ịzụlite na-adịghị mma mgbaàmà ndị dị otú ahụ dị ka dizziness, isi ọwụwa na ịmụ anya arọ nrọ. Ke adianade do, anyị na-apụghị ewepu paranoid omume.
Na ovadozu emetụta saa afo na symptomatic ọgwụ.
bụ dakọtara na ndị ọzọ ọgwụ ọjọọ eme ihe
Imekotaotuugbo ngwa nke ihe ngwọta na mbadamba "Futsis" na anticoagulants budata amplifies mmetụta ha. Ya mere, na-aga n'ihu nlekota nke egosi nke prothrombin oge.
Weere na nkà mmụta ọgwụ nwere ike dịkwuo plasma kasịnụ nke "benzodiazepines", "Midazolam", "Cyclosporin", "phenytoin" na "rifabutin" ke iyịp. Flucanozole Mgbe jikọtara ọ bụla n'ime ndị a n'aka na-achọ dose mgbanwe na chọpụtara nwere ọkachamara. Ọ bụrụ na anyị eleghara ndụmọdụ data, dị n'ịgwa nwere ike dịkwuo mmetụta nke psychomotor Jeremaya mere akpata mmepe na na.
Na mgbe nile were nke hydrochlorothiazide na "Futsisom" i nwere ike na-atụ anya a ịrịba ama mmụba na ọbara ịta nke fluconazole. Otú ọ dị, nke a adịghị achọ a dose ukpụhọde.
Ịnata kwuru ọgwụ adịghị belata ihe nke jikọrọ ọnụ na gbochie afọ.
The ọgwụ "Futsisom" Ọrịa na-arịa ọrịa shuga kwesịrị ichebara puru omume mmepe nke hypoglycemia.
Imekotaotuugbo ọgwụgwọ na a ọgwụ, "rifampicin" na-achọ onye na-abawanye na dose of fluconazole.
The Nchikota "Futsisa" na "Tacrolimus" ọtụtụ mgbe na-akpata ibe nkwalite nke ha nephrotoxicity.
Na-eri na analogues nke ihe antifungal gị n'ụlọnga
Ịgbaso nhọpụta nke "Futsis" antifungal ọgwụ, ọtụtụ ndị ọrịa na-ajụ banyere otú ọ na-efu. Ọ ga-kwuru na price nke ọgwụ na dị iche iche na-ere ọgwụ ígwè nwere ike iche ubé. Ya nkezi na-eri bụ banyere 300-400 rubles (n'agbanyeghị ụdị ntọhapụ).
N'ihi na ọgwụ ọjọọ, yiri na pharmacological e ji mara na-agụnye ọgwụ ndị dị otú ahụ dị ka "Fluconazole", "Fukortsin", "Clotrimazole" na "Livarol". Otú ọ dị, na ha n'ikuku kwesịrị maara na ha nwere ike a kpamkpam dị iche iche mmetụta na contraindications. Ya mere, i kwesịrị mgbe ịkpọ onye dọkịta na-eji dochie "Futsisa" site ndị a n'aka. Site n'ụzọ, nke ikpeazụ ga-enwe ike eburu gị maka ezi na kasị dị irè ọgwụgwọ Usoro.
Nleba nke antifungal mmadụ
Ọtụtụ mgbe atụle a nkwadebe maka ahapụ mma nzaghachi. Dị ka ọhụrụ, ọ na-ezi ọtụtụ-eji gynecological omume na ọgwụgwọ nke thrush. Otú ọ dị, ọtụtụ ndị na-arụ ụka na-emegide fungal gị n'ụlọnga "Futsis" na-enyere tufuo a wetara ọrịa n'ihi na ezi a ogologo oge. Otú ọ dị, ndị ọkachamara na-akọ na otu onye na-ekwesịghị ichefu banyere ọgwụ ndị ọzọ na-eme ka ndị nkịtị na osisi na ikpu.
Na-ekwu okwu banyere ịdị irè nke "Futsis" ọgwụ ọjọọ, ghara ikwu ihe ọjọọ nzaghachi. Ụfọdụ ọrịa emeso ya na a ọgwụ, na-ekwu na oriri nke mbadamba ma ọ bụ ojiji nke ngwọta na ha hụrụ mmetụta. Dị ka a na-achị, ha na-egosi ọzịza, itching, mucous membranes nke imi na anya, ahụ ọkụ, na oké isi ọwụwa.
Amaedi "Futsis" jel, na reviews banyere ya bụ ihe na-erughị nkịtị. Na ndị na-, dị ka elu arụmọrụ nke a na-ajụ, karịsịa na ọgwụgwọ nke tinea.
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