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Analogue "Diflucan" - pụtara "Fluconazole"

Analogue "Diflucan" - pụtara "Fluconazole" - bụ ihe antifungal gị n'ụlọnga na-enwe a ukwuu kpọmkwem mmetụta. The ọgwụ ike igbochi ọrụ nke ụfọdụ enzymes, inhibit mgbanwe nke lanosterol ka ergosterol. Ke adianade do, ọgwụ enwekwu permeability nke cell membranes, na-egbochi replication na uto nke pathogens. The ọgwụ dị irè maka opportunistic fungal-efe efe iwe na fungi genus Candida, gụnyere generalized immunosuppression ụdị candidiasis ke ala. Na Ịṅụ ọgwụ nwere ezigbo absorbability. Na ọnụego nke absorption na-adịghị emetụta nri oriri. The bioavailability nke ọgwụ bụ banyere 90%. Oke ọdịnaya ọbara esịmde a na-agwọ na 30-90 nkeji. The ọgwụ na-ọma na-ekesa na nsụkọrọ na oke mmiri banye n'ime n'ime mmiri ara ehi. Ọ ga-kwuru na price nke ọgwụ "Fluconazole" iwu nke ịdị ukwuu ala karịa uru nke "Diflucan" (n'oge gara aga ga-akwụ site na narị anọ na narị asatọ rubles).

na-agba akaebe

Medicine "Fluconazole" (analogue "Diflucan") na-kenyere na cryptococcal meningitis, cryptococcosis na ndị ọzọ na localizations cryptococcal ọrịa ọrịa na a nkịtị dịghịzi omume na na dị iche iche nke immunosuppression. Site àmà nke candidiasis gụnyere generalized ụdị, akwadebe candidiasis, candidemia, na ndị ọzọ ụdị invasive efe efe mere site a ero Candida. The na nkà mmụta ọgwụ na-atụ aro maka mgbochi nke fungal-efe efe na ọrịa na ịza aza etuto ahụ nke agwa. E Kenyere gị n'ụlọnga maka mycosis ụkwụ, ukwu, toso.

dosing Usoro

Analogue "Diflucan" - pụtara "Fluconazole" - kenyere ka ọrịa na afọ iri na ise na a uka ukwuu karịa 50 n'arọ. Mgbe cryptococcal na-efe efe nke dị iche iche orunótu n'ubọchi mbu na a dose nke 400 mg. Gasịrị, ego nke agwọ ọrịa belata ka 200 mg kwa ụbọchị. Duration nke ọgwụ ndị a na pathologies na-adabere na arụmọrụ nke ọgwụgwọ, nke na-egosi na mycological ọmụmụ. Ngwa nke cryptococcal meningitis ga-adịru dịkarịa ala isii na asatọ izu. Mgbe akwadebe candidiasis, candidemia, na ndị ọzọ ụdị invasive Candida na-efe efe n'ụbọchị nke mbụ ego nke ọgwụ - 400 mg, na onunu ogwu na-ebelata ka 200 mg. Bụrụ na nke ezughi oke irè nke ọgwụgwọ na onunu ogwu na-ụba azụ 400 mg. Na oge nke ọgwụgwọ na-adabere na irè nke n'aka.

n'akụkụ mmetụta

Analogue "Diflucan" - ọgwụ "Fluconazole" - nwere ike ime ka dizziness, ihe mgbu na isi, afo, abdominal mgbu, ogbenye agụụ, ọgbụgbọ. Na ndabere nke ọgwụgwọ nwere ike ịzụlite thrombocytopenia, nfụkasị Jeremaya dị ka ọzịza nke ihu, epidermal nsí necrolysis, akpụkpọ itching. Analogs mbadamba nwere ike ime ka emeghasịkwa nke imeju, akụrụ, hypokalemia, hypertriglyceridemia.

contraindications

Ekwela idepụta ọgwụ tupu afọ 4 afọ, bụrụ na nke ekweghị ibe nọrọ nke ya mmiri. Contraindicated jikọtara eji na agwọ ọrịa "Terfenadine", "Astemizole" na ndị ọzọ so na ogologo oge QT-nkeji. Ịkpachara anya n'oge ọgwụ na show pụrụ ịrịa dị iche iche pathologies (na electrolyte ahaghị nhata, organic ọrịa obi na ọrịa, wdg).

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