Ahụ ike, Preparations
Aromatase inhibitors: reviews, ahịa. Aromatase inhibitors na bodybuilding
Aromatase inhibitors, ma ọ bụ blockers, - ụdị agwọ ngwaọrụ na-eji belata ịta nke estrogen n'ime ọbara na-amụba na ọkwa nke gonadotropins na testosterone. Ndị bekee na-eji maka ọgwụgwọ na mgbochi nke nwoke gynecomastia.
Aromatase inhibitors na bodybuilding na-eji n'oge N'ezie nke Steroid anabolic to:
- melite arụmọrụ nke anabolic homonụ na ọbara;
- gynecomastia mgbochi;
- gbochie ọbara mgbali;
- dịkwuo okuku (site na iwepu mmetụta ọjọọ n'ahụ nke estrogens);
- mbenata estrogen mbibi axis testicles-pituitary-hypothalamus, nke na-eduga ná a na-awụ ọsọ nwughari.
Iwuli a N'ezie, ị ga-ewere ya na eziokwu na flavor bụ n'okpuru niile anabolic Steroid. Iji na-agu n'onye ezi omume mgbe ojiji nke ngwaahịa ndị dị otú ahụ dị ka methandrostenolone, methyltestosterone, testosterone na-eji ya emepụta. Ubé flavored Halotestin, boldenone.
irè
Ndị kasị họọrọ na dị aromatase inhibitors (n'ihi na na-amị mkpụrụ fọrọ yiri):
isiokwu (Global aha) | Brand (rere site pharmacies) | ndika price | ntọhapụ Ụdị | prophylactic bodybuilding | Mgbe gynecomastia |
"Exemestane" | "AROMASIN" | 1600 ete. | 30 Tab. 25 mg | 2.5 mg (ọkara mbadamba) kwa ụbọchị | 25 mg kwa ụbọchị ruo mgbe mgbaàmà liquidation. Mgbe onunu ogwu Mbelata ka prophylactic. |
'Letrozole' | "Letromara" (Farmak). "Letroza" "Estrolet" | 3200 rubles. 1000 rubles. | 30 Tab. 2.5 mg | 0,5 mg (1/5 mbadamba) kwa ụbọchị | 2.5 mg kwa ụbọchị ruo mgbe mgbaàmà mkpochapu. Mgbe onunu ogwu Mbelata na mgbochi. |
"Anastrozole" | "Village" "Egistrazol" "Anastrozole Kabi" | 1500 rubles. 350 rubles. 1300 rubles. | 28 Tab. 1 mg | 0,5 mg (ọkara mbadamba) kwa ụbọchị | 1 mg kwa ụbọchị ruo mgbe mgbaàmà liquidation. Ọzọkwa Mbelata ka prophylactic onunu ogwu. |
Ọ ga-kwuru na a agafeghị oke ịta nke estrogen bụ bara uru n'ihi na muscle ibu, ọ dị preventative Dosages gosiri na quantities emetụta ichebe physiologically chọrọ larịị nke nwoke estrogens.
Iji N'ezie
Ihe ka ọtụtụ n'ime anụ ụlọ na-eme egwuregwu na-eji aromatase inhibitors, iji na-eso eme: ọgwụ ọjọọ na-eji naanị mgbe mbụ ihe ịrịba ama nke gynecomastia (itching nke nipples, ọzịza, nācha ọbara-ọbara). N'ụzọ dị mwute, a na-enweghị ike na-akpọ ezigbo.
The kasị ò ngwọta na-atụle-anwale estradiol na banyere ụbọchị iri, na ojiji nke anabolic Steroid na a obere ọkara ndụ ( "Methandrostenolone", "Testosterone propionate") ma ọ bụ atọ ma ọ bụ anọ na izu nke ngwa nke elongated Ester ( "Sustanon", "enanthate," "cypionate"). Ọzọkwa kenyere nkezi òkè "Anastrozole" - 0,5 mg kwa ụbọchị. Mgbe ụbọchị iri, ẹkenịmde a ịchịkwa analysis of estradiol na onunu ogwu na-gbanwee dị ka na-arụpụta.
Ikwere bụ iji ala na-agafeghị oke servings "Anastrozole" lekwasịrị anya onye amụta. Ọ bụrụ na mgbe dị otú ahụ a ọgwụgwọ na-aghọ ndị dara mbà n'obi, aghara nke erectile ọrụ, libido dobe, mgbe ahụ ị chọrọ iji belata dose.
research
Ntoputa nke a n'ihu ọha ika "letrazole" ada ngwaahịa a n'ime ndú. E nwere a dịgasị iche iche nke ule iji gosi na elu irè nke ngwá ọrụ a na ndị ikom. The mmeghe nke bekee esonyere a nnọọ ịrị elu nke gonadotropin (LH). Arụpụta onunu ogwu, si n'aka si 0,02 mg (ọgwụgwọ n'okpuru 100 ugboro): ọ bụ omume na via a atọ ala estrogen ịta. 50% "letrozole" tutu amama si ahụ n'ime 2-4 ụbọchị, ka o wee na-aṅụ a ụbọchị. Ihe bụ isi drawback-atụle ga-ike ka ala etoju nke estrogen, ọbụna obere doses.
"Anastrozole" na-ewu ewu na bodybuilding, ya ịrịba ama na-amụ na ndị dị ka a n'aka mbenata estradiol. Empirically ọ e gosiri na a dose nke 1-0.5 mg estradiol ozo nwere ike ibelata site dị 50%. Na-ere ahịa Ngwaahịa a nwere ike zụrụ ruo ugboro iri dị ọnụ ala karịa ahịa ọgwụ. Na megacities osobo cheap "Anastrozole Kabi."
N'akwụkwọ ya, Dr. Mauro G. De onwa dere, sị: "Ọ na-chere na estrogens na-guzobere n'ihi nke aromatization nke testosterone ma ọ bụ ndị ọzọ anabolic Steroid na ngalaba nke hypothalamus na ụbụrụ, na-ebelata secretion nke luteinizing hormone, na, mmọdo, na mmepụta nke testosterone." Gilman na Goodman asian na nzaghachi na-arụ ọrụ kama ihe ìgwè estrogen, kama testosterone. N'ụzọ dị otú a, ọ na-kọwara na aromatase inhibitors nwere ike budata belata inhibitory mmetụta nke anabolic mmadụ igbunye onye mmekọahụ homonụ.
mmetụta
The aromatase inhibitors ndị dị ize ndụ nke ndị ikom? Anyị maara na estrogen na ala doses nwere nti utịp ke nwoke ahu. Estrogen homonụ dịkwuo na dịruru arụmọrụ na uche nke androgen anabata. Ọzọkwa, ha onwe ha nwere a nchebe na anabolic mmetụta.
Pụtara muscle estrogen ihe nnabata juputara kọwara Anna Wiik na zuru ezu. N'ezie-akpali mmasị n'ezie blocker dose nwere ike isi ibelata estrogen, nke na-eme ka ntoputa nke mmetụta ndị dị otú ahụ dị ka:
- mgbochi nke muscle ibu;
- nkwonkwo mgbu (arthralgia);
- ahụ ike na-arịa ọrịa na iju ke libido;
- ịda mbà n'obi;
- aghara nke ọbara lipid profaịlụ (cholesterol abawanye);
- ibelata na ọkpụkpụ ike.
Subjectively, ọgwụ ndị mma anabata karịa "Tamoxifen".
eke inhibitors
Na-na-esonụ:
- caffeine;
- resveratrol;
- zinc;
- nicotine;
- apigenin;
- catechins;
- eriodiktiol.
The iji "Anastrozole"
More karịa ezi aromatase inhibitors? ọgwụ ndị a na-ọtụtụ-eji bodybuilding. Ka ihe atụ, "Anastrozole" chọrọ maka mmiri njigide na ahụ mmadụ na mgbochi nke omume nke gynecomastia (mgbe na Nchikota na androgens testosterone na Dianabol ụdị ma ọ bụ na Nchikota na finasteride). Ma na nke a, ndị na-eme egwuregwu na-akawanye na nnukwu mgbagwoju nke machibidoro iwu ọgwụ ọjọọ si "ndepụta iwu bekee na ụzọ", e wezụga na-enwe ya nso nke abụọ mmetụta.
The na-achịkwaghị achịkwa ojiji nke "Anastrozole" na-eme egwuregwu, na-ebu banyere, akpan akpan, bodybuilding nwere ike ime ka arthralgia, asthenia, ma ọ bụ iji belata agagharị nke nkwonkwo, isi ọwụwa, somnolence. N'ezie, mgbe ụfọdụ nwere ike na-egosi thromboembolic nsogbu na ịzụlite ọnụ ụtarị.
On "Anastrozole" Ọtụtụ e dere akwụkwọ maka na-eme egwuregwu dị ka a nnọọ na-adịghị njọ ọgwụ. Ma anya na ozugbo mmetụta na ya n'ikuku pụrụ ịbụ nnọọ na-ejighị n'aka na mwute. N'ezie, ọ bụrụ na naanị otu mbadamba (1 mg) kwa ụbọchị, nwere ike kwadebere akpọ hormone anya. Site n'ụzọ, a onu a hụrụ na ihe karịrị 80% nke ndị na-eji ngwaahịa.
Ke ofụri ofụri, aromatase inhibitors - ọgwụ ọjọọ mara ezuru. amụba atọ samples blockers "Anastrozole", na mgbe e mesịrị "vorozole" na
'Letrozole', e kere dị ka ngwaahịa nke mbụ na nke abụọ edoghi na-agwọ ọrịa gbasasịa ihe nnabata-mma ara cancer.
"Krizin"
N'ihi weightlifters pharmacological ahịa nakwa awade a 5.7-digidroksiflavon ( "Krizin"), nke na-eme egwuregwu na-eji na nnọọ elu doses. Ọ nwere antiaromatazatnymi Njirimara na-emepụta abụọ forms - MRM-Chrysin, nyere 500 mg kwa Capsule enweghị ntụpọ krizina na SciFit-Chrysin Njedebe, nyere ọkara ifịk umi.
Mmetụta nke na mmepe na-igosipụta, ma ọ ga-eti na niile bekee na preparations enwe antiaromatazatnym edinam, ike nke na-eme ihe ọjọọ ahụ otu nnukwu na-eme egwuregwu. Ọzọkwa, ha na-na "Ndepụta nke machibidoro bekee na ụzọ."
Nyocha
Ọtụtụ bodybuilders na-ekwu na, dabere na ahụmahụ na "letrozole" ( "Femara"), ha kwubiri, sị: Ngwaahịa a, site idozi otu nsogbu (elu egosi estrogen), na-akwalite ntoputa nke ọtụtụ nsogbu ndị ọzọ. N'ezie, aromatase inhibitors dị mkpa maka ndị ikom. Mgbe niile, ndị ahụ (ndị ikom na-akpan akpan) eji estrogen iji chebe ahụ ike nke dịghịzi usoro, ụbụrụ, nkịtị cholesterol etoju, nkwonkwo, ụdọ, na na.
Na-eme egwuregwu na-ekwu na estrogen akpali ahụ usoro nke muscle ibu. Inweta 2,5 mg "letrozole" n'ụbọchị ha na-amalite na-eche oké njọ mmerụ articular nkwonkwo na akwara njikọ, ma na-enweghị ka na-efe efe na malitere ịrịa ọrịa na.
Ọtụtụ na-eme egwuregwu kwere na 'Letrozole' ike ga-eji naanị ọkachamara bodybuilders na nkwadebe maka agbụrụ. N'ihi ya, ha tufuo ngafe ọmụmụ na ahu (maka ndị ọkachamara ahụ ike n'ihi na mmeri bụ ndo). Ha nwere obi ụtọ-na aromatase inhibitor. Ha price bụ nnọọ afọ ojuju.
Ụfọdụ na-eme egwuregwu na-ekwu na 'Letrozole' mmetụta dị mma n'ahụ ọbụna na a dose nke 0.1-0.5 mg. Ha na-akọ na ọ bụghị njọ karịa obere mmetụta nke ndị ọzọ inhibitors, na ọkọlọtọ maka nke a ụdị ọgwụ. Ha na-ekwu na subjectively, ngwaahịa na ngwa ngwa revolutionizing testicular olu karịa "Tamoxifen" na "Clomid". Ha na-arụ ụka na aromatase inhibitors - ọgwụ ọjọọ eme ihe na-eri di mma.
Ụfọdụ na-eme egwuregwu akụkọ na ike ga-eji ọ bụla blocker, ma nyere elu arụpụtaghị "letrozole" na obere doses, ọ bụ ihe kasị ọnụ.
"Anastrozole"
Taa "Anastrozole" bụ ndị kasị ewu ewu blocker. Ndị dị ọnụ ala a na-ewere na "obodo." Ụfọdụ n'ime aromatase inhibitors na ahịa ọgwụ na-obere, n'ihi na ihe atụ, "Anastrozole Kabi."
Ọtụtụ ndị adịghị azọpụta na ahụ ike ha na-ahọrọ na-mma.
Were "Anastrozole" dị na ya dị larịị nke estradiol. Ya mere mbụ na-anwale estradiol etoju ịgbanwe dabeere na analysis òkè. Nkezi oge gboo onunu ogwu bụ 0,5 mg kwa ụbọchị.
Mgbe ụbọchị iri gasịrị, mkpa ka i ina-anwale ọzọ. Ọ bụrụ na larịị nke estradiol a ọkọlọtọ, ọ bụ ike iji belata onunu ogwu nke 0,5 mg ugboro abụọ n'izu. Ọ bụrụ na ọ bụ ka elu, n'ikuku ga-aka iso. N'ihi ya, ọ ga-abụ na mmetụta ruo mgbe zuru mgbake estradiol etoju.
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