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"Clonazepam": reviews. "Clonazepam": ntuziaka maka ojiji, mmetụta

"Clonazepam" - antiepileptic ọgwụ nke na-akọ ka benzodiazepine emepụta. Mgbe e ndị "clonazepam" Fim na-ekpe na-akasị mma iji ọgwụ. The ọgwụ nwere muscle relaxant na ogwuura mmetụta, ma na-nwere a ogwuura mmetụta.

The mejupụtara, ntọhapụ ụdị "clonazepam" ọgwụ

The ọgwụ dị na mbadamba na dị iche iche ọdịnaya nke isi mmiri:

  • 0,5 mg. Ke adianade clonazepam, Ọdịdị na-agụnye lactose monohydrate. Iji Efrata nke mbadamba na-emetụta sodium carboxymethylstarch. "Clonazepam" mbadamba nwere magnesium stearate, gelatine. Auxiliaries nwekwara talc na nduku starch. Agba mbadamba mmasị e ji esiji ákwà E110.
  • 2 mg. Ọzọ inyeaka Efrata - polysorbate 80, lactose monohydrate. The mejupụtara nke ọgwụ ugbu carboxymethylstarch sodium na sodium lauryl sulphate. talc, gelatin bụ ịnara Efrata. Inyeaka mmiri ma nwe ọzọ bekee - magnesium stearate, osikapa, nduku starch.

Pharmacological edinam "clonazepam" ọgwụ

"Clonazepam" a nkụda mmụọ na a ọnụ ọgụgụ buru ibu nke owuwu na-eme ka Central ụjọ usoro, tumadi na ndị na-na-metụtara obi ịrụ ọrụ. Mmetụta nke ọgwụ ọjọọ, "clonazepam" ntụziaka ntuziaka, nzaghachi egosipụta ka a ogwuura, anxiolytic na hypnotic (ikpeazụ moderately owụt). The agwọ ọrịa ebelata skeletal Akwara ụda, na-egbochi generalized convulsive ọdịdọ. E nwere a mmetụta dị mma na N'ezie nke akwụkwụ ọgụ (Baịbụl hiwere isi n'ebe, generalized).

Pharmacokinetics

The ọgwụ na-fọrọ nke nta kpamkpam etinye obi gị dum na eriri afọ tract na-outputted tumadi site na akụrụ (metabolites), a obere akụkụ (2%) na-egosi na-agbanweghi agbanwe. The usoro na-ewe a ọkara ndụ nke 20 na 40 awa. The bioavailability nke ingested nkwadebe bụ 90%, na mmekọrịta ya na ọbara ọkọnọ - 85%, nke kachasi elu ịta ruru a pụtara nke 2.5 awa. Na ọgwụgwọ nke "clonazepam" ya mmiri ga-esi n'ime mmiri ara.

Egosi maka ojiji nke ọgwụ

Mbadamba "clonazepam" kwesịrị ekwesị n'ihi na ọgwụgwọ nke ọrịa dị iche iche afọ na Akwụkwụ na-adọ, n'agbanyeghị ya ngosipụta:

  • ele mmadụ anya n'ihu ihe ọdịdọ (obodo, Baịbụl hiwere isi n'ebe) nke ọ bụla ogo ogo;
  • convulsive ọnọdụ (tonic, clonic);
  • mfe ọdịdọ nke abua generalized;
  • gbara gharịị abịaghị (Lennox-Gastaut syndrome);
  • myoclonic ọdịdọ;
  • ahụkarị enweghị ọdịdọ;
  • tonic-clonic ọdịdọ isi na sekọndrị pụta ìhè.

"Clonazepam" kenyere iji belata muscle ụda, ma hypnotic na psychomotor ọdụdọ n'oge ọgwụgwọ.

The iji ọgwụ ọjọọ eme "clonazepam"

The chọrọ onunu ogwu kpebisiri ike dabere na ọtụtụ ihe. Mgbe mbụ ogbo nke ọgwụ na-eji a obere dose "clonazepam" (0,5 mg), ji nwayọọ nwayọọ na-agbanwe agbanwe na onunu ogwu ruo mgbe mkpuruedemede mmetụta na-enwetara. N'otu oge gafere karịa onunu ogwu a ka amachibidoro. Dị ka reviews, "clonazepam" enweghị ike inikiet inikiet weliri ọbụna mgbe ọgwụgwọ adịteghị. Nkọ ojuju nke ọgwụ egwu mmepe nke onye akwụkwụ, ọnọdụ ọdịdọ.

Admission Akwụkwụ na-adọ:

  • Okenye. Mbụ ọgwụ na-rụrụ iji karịa 1 mg nke ọgwụ. The dose gbakọọ kwa ụbọchị, kewara 3 ma ọ bụ 4 doses, nke a ga-rụrụ na mgbe etiti oge. Enweghị ikike iji ọgwụ ke hà doses, ndị kasị ibu òkè nke "clonazepam" ọṅụṅụ tupu na-aga ụra. A, zuru ezu kwa ụbọchị onunu ogwu bụ na nso nke 4 ka 8 mg ọgwụ. Mmezi dose ekwesịghị gafere 20 mg (enweta n'oge 2-4 izu nke ọgwụ). Mgbe kpebisiri ike irè kwa ụbọchị dose, nke na-enye ohere ịnọgide na-enwe nkịtị ọnọdụ nke ahụ, ọ na-ekwe ka otu dose na alakpu ụra.
  • Children (site na ibu ibu nke dịkarịa ala 30 n'arọ). Dị ka reviews, "clonazepam" na mbụ gosiri maka ụmụaka 0,5 mg iji chọpụta ya ezigbo dose.

N'ikuku na syndrome, nke na-esonyere paroxysmal mgbu:

  • Okenye. Akpa, na ọrịa na-ndinọ 1-2 ụbọchị dosing (0,5 mg oge ọ bụla). Ọtụtụ ndị ọrịa zuru ezu ọgwụgwọ dose bụ 1 mg / ụbọchị. The ụbọchị ike na-aṅụ ihe karịrị 1 mg nke ọgwụ ọjọọ, "clonazepam". Nyocha, Otú ọ dị, na-egosi na n'ọnọdụ ụfọdụ, ndị dọkịta pụrụ ịmụba dose 4 mg. N'ọnọdụ dị otú ahụ, na onunu ogwu na-eji nwayọọ nwayọọ gbanwere (nso - 3 ụbọchị, ikekwe na-agbakwunye 0,5 mg). Mgbe ị chọrọ iji belata ogo ụra n'ehihie, na dose gbakọọ na n'ikuku n'ụbọchị, i nwere ike na-aṅụ tupu alakpu ụra.
  • Children. N'ihi na ọrịa ndị na-adịghị okenye karịrị afọ 18, nchọpụta nke syndrome ọgwụ nwere ike na-adịghị ike na nwedịrị ike ịta.

Iji zere ihe ọ bụla nsogbu, ọgwụ "clonazepam" reviews nke dọkịta nwere ike ikwu na-ewere nnọọ na-atụ aro nke a ọkachamara na-na-emeso.

Contraindications inweta "clonazepam" ọgwụ

Mbadamba na-agaghị eji mgbe ụba uche na bekee site nke ha na-ekewet. The ọgwụ na-contraindicated na ndị a na-ekwu:

  • myasthenia gravis;
  • impairment nke nsụhọ;
  • n'ịmụ nwa, ara;
  • glaucoma (mmechi);
  • akụkụ okuku ume na ọrịa na-enwe a Central si malite, oké akụkụ okuku ume na insufficiency;
  • Arọ aga gbasara akụrụ na hepatic ọdịda;
  • ngosipụta nke ụra apnea syndrome;
  • mmanya nsi;
  • porphyria nnukwu ụdị.

Mmetụta "clonazepam" ọgwụ

Tụlee mmetụta, nke nwere ike ime ka "clonazepam". Iji ọgwụ ike ga-metụtara oghom Jeremaya mere. Nwere ike ime ka lethargy, ọgbụgbọ, ahụ mgbakasị. Ọ bụrụ na ihe oghom mmeghachi omume site ahụ mmadụ ego n'anya ike gwụ ngwa ngwa, ọ nọwo na nchikota nke mmegharị. Iji belata mmetụta nke ediyarade nke mmetụta, mbụ ị mkpa itinye a obere dose, jiri nwayọọ nwayọọ na-amụba ruo mgbe ọ na-aghọ ezigbo.

Ọ maara na n'oge ọgwụgwọ "clonazepam" pụtara iji ya na mebiri nke na-atụ aro nwere ike ime ka ovadozu. N'ọnọdụ dị otú ahụ, e nwere a pụtara, bụ nke pụrụ iduga aghara, stupor, nke nwere ike ịkpata a amaghị onwe ya. Tinyere ihe ndị ọzọ mgbaàmà - vaskụla ida, mkpọchị ume, iro ụra. Ọ dị mkpa na-asa na afo (irè ozugbo ewe mbadamba) kụziere kwesịrị ekwesị ọgwụ. Ọ dị mkpa ka mgbe niile nyochaa mgbanwe egosi ndị dị otú ahụ dị ka ọbara mgbali, usu, iku ume. Mgbe ụfọdụ, ọ na-achọ mmejuputa n'ibu ventilashion. E nwere ihe ngwọta - "Flyumazenil," ma ọ bụ adabara ochichi ka ọrịa a na-na-emeso "clonazepam" ruo ogologo oge.

Ọ dịghị mkpa ka ikpokọta "clonazepam" na-aba n'anya. Nyocha ekwe iji jide n'aka na ndị dị otú a Nchikota nwere ike inwe ihe ize ndụ ndụ. The otu na-emetụta niile ọgwụ ọjọọ na-eme ihe na Central ụjọ usoro, inhibiting ọrụ ya.

Drug mmekọrịta "clonazepam" nkwadebe

Mmetụta nke ọgwụ dịkwuo narcotic analgesics, anticonvulsants. Otu N'ihi a hụrụ site na ijikọta ya antidepressants, neuroleptics, barbiturates, nakwa mgbe jikọtara na mmanya na bekee ebelata skeletal Akwara ụda. Irè nke ọgwụgwọ na-ebelata mgbe ingested nicotine.

Na-eri, reviews banyere ọgwụ ọjọọ, "clonazepam"

Zụrụ "clonazepam" mkpụrụ ọgwụ na Moscow nwere ike ịbụ n'ihi 97-150 rubles. (30 PC.). The ọgwụ bụ irè Akwụkwụ na-adọ, ma ọ bụrụ na kwetara na a dọkịta nkwanye. Mgbe atonic ọdịdọ nwere ike ọnwa abụọ, oge nke ọgwụ bụ zuru ezu maka ndị dị otú ahụ a oge, ị nwere ike ịgbanwee mmezi ọgwụgwọ. Mgbe ụfọdụ, e nwere mmetụta, ma ukwuu n'ime naanị na mbụ na-adọ ọgwụgwọ, mgbe mgbe, a adịghị ike.

Ikpe ikpe site ọmụma na-ebu reviews, "clonazepam" ego n'anya Bibie nke ụba Akwara ụda na banyere izu atọ. Dọkịta nwere ike nye iwu ka ọgwụ na ikpe nke na oti mkpu, egwu, IRR, nke na-esonyere egwu ọgụ. The ọgwụ dị irè, na-arụ ọrụ ngwa ngwa.

Nyocha "clonazepam" na-egosipụta dị ka a ọma n'aka na-eme ya ọrụ, ma nwere ike ime ka nsogbu ahụ ike (adịghị ike, ike ọgwụgwụ, na na. P.).

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