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Codeine phosphate: ntuziaka maka ojiji, analogs na reviews

Codeine bụ nke ọgwụ opium alkaloids usoro. Ọ na ọtụtụ-eji nkà mmụta ọgwụ dị ka a usọbọ maka ụkwara. Ọ na-ezo aka a centrally eme ọgwụ nke a na-eji na Nchikota na ndị ọzọ bekee, otu nke bụ terpin hydrate. Ezi na-akpali bụ eziokwu na ojiji nke codeine pụrụ igosipụta ihe ịrịba ama nke ọgwụ mmenaanya. Kwuru, na analgesic mmetụta. Na nke a, codeine phosphate ike ga-eji dị ka ihe mgbochi ụfụ, kama nditịm site ọgwụ.

nkenke ọmụma

Ụkpụrụ nke ime ihe dị yiri nnọọ codeine ka morphine. Otú ọ dị, ya analgesic mmetụta ndị dịtụ na-adịghị ike. Ọnụ na a codeine phosphate (Latin na-egosi a umi dị ka codeinum) nwere ike akpọ ike belata excitation ụkwara center. Ịga n'ihu ntụnyere na morphine, ihe atụ, na ọ bụ nnọọ obere mwute mmadụ ume, na ọ bụghị nke ukwuu na-egbochi ọrụ nke eriri afọ tract. N'agbanyeghị nke a, ezi mgbe e nwere otu ebe ọgwụ nwere a na-akpali akpali mmetụta na ozu, na-egbochi iro ụra.

Codeine phosphate: nkọwa contraindications

Dị ka ndị ọzọ ọgwụ, codeine nwere otu nnukwu ndepụta contraindications. Ha ga-hoo haa mara tupu ị na-eji eri. Iji mma gị na nghọta, anyị na-anọrọ ha na a iche iche na ndepụta. N'ihi ya, ọgwụ na-ekwesịghị-eji na ọnụnọ nke ndị na-esonụ ihe:

  • High hypersensitivity;
  • arrhythmia;
  • igbu onwe;
  • nsia nsogbu, prostate gland na urethra;
  • ime ma ọ bụ lactation;
  • agadi ma ọ bụ ụmụ afọ;
  • Dabere na nnweta nke ọgwụ umi akpọ codeine phosphate;
  • afọ ọsịsa;
  • nsogbu na aṅụrụma;
  • na-egbu egbu dispensiya;
  • ọnụnọ nke mwakpo nke bronchial ụkwara ume ọkụ;
  • mmerụ ahụ n'ụbụrụ, nakwa dị ka akụrụ ma ọ bụ mmebi imeju.

Dị ka ị pụrụ ịhụ, na ndepụta bụ nnọọ nnukwu. Ke ofụri ofụri, tupu ojiji nke codeine kwesịrị bụchaghị ịkpọ dọkịta gị. Ọ ga-nye iwu ndị dị mkpa ọgwụ ma ọ bụrụ na ọnọdụ ahụ gị-enye gị ohere-a na nkà mmụta ọgwụ.

Codeine phosphate: otú na-na na ihe doses?

Mgbe na-eji codeine maka ọgwụ nzube kwesịrị karịsịa ịkpachara anya mgbe drafting ziri ezi onunu ogwu nke umi, nakwa dị ka oge nke ya mbanye. Ya mere, bụrụ na nke nnukwu mgbu ọ na-atụ aro n'ihi na ndị okenye na-15-60 mg ọ bụla 3-6 awa. Mgbe afọ ọsịsa na-ebelata ka a onunu ogwu nke 30 mg anọ ugboro n'ụbọchị. N'ikpeazụ, mgbe ụkwara ọdịdọ ga na-aṅụ 10-20 mg nke ọgwụ 4 ugboro n'ụbọchị. Higher kwa ụbọchị dose of codeine phosphate nke (nwere dee a ọgwụ dọkịta) bụ 120 mg.

N'ihi na ụmụ nke usoro onunu ogwu a obere bit dị iche iche. A, ruru bụ nke 0,5 mg kwa 1 n'arọ nke ahu arọ, mgbe ọ na-abịa n'igbochi iche iche mgbu. Mgbe ị na ụkwara ị na-ekwesịghị-ewe ihe karịrị 15 mg. N'ikpeazụ, na afọ ọsịsa ka na onunu ogwu bụ 0,5 mg kwa 1 n'arọ nke ahu aro. Banyere ugboro nke n'ikuku, ọ bụ, dị ka okenye, ga-hà 4-5 ugboro n'ụbọchị. Site n'ụzọ, ụmụ n'okpuru anata codeine phosphate adịghị atụ aro 2 afọ.

pharmacological mmetụta

Dị ka e kwuru na mbụ, codeine bụ a centrally eme antitussive. Ọ bụ nke phenanthrene alkaloids nke usoro. Ọzọkwa, ọ na-akọ opioid ihe nnabata agonists na pụrụ n'ụzọ dị ukwuu belata excitability nke ụkwara center, ruru ya kpọmkwem mgbochi. Ịnụ ọgwụ ọrụ pụrụ ịkọwa umi ebighị nke opiate anabata na igosipụta excitation na ọtụtụ akụkụ nke Central ụjọ usoro. Plus, ọ na-na-agbanwe ọnụ ọgụgụ nke obi nghọta nke ihe mgbu. N'ozuzu, ndị analgesic mmetụta na-egosipụta onwe ya mgbe 10-45 nkeji mgbe ogwu ogbugba, na via ọkara otu awa mgbe eji codeine phosphate mbadamba. Na oge nke edinam dịruru ihe 4 awa.

mmetụta

N'ezie, codeine phosphate nwere ya mmetụta, nke onye ọ bụla nwere ike na-egosipụta n'ụzọ dị iche iche. Dị ka n'ihe banyere contraindications, anyị na-enye ndepụta nke mmetụta na-egosipụta onwe ha mgbe iji nke a umi:

  • The ụjọ usoro nwere ike dị otú ahụ gbuo edinam: ụba iro ụra, isi ọwụwa na dizziness (obere), ekwe omume nke ịmụ anya arọ nrọ ma ọ bụ visual mmegharị anya, nchegbu, na-arọ nrọ n'ime nrọ, ịda mbà n'obi (a obere omume), nakwa dị ka ihe ọdịdọ. Mgbe oriri nke oké doses nwere ike mara jijiji, na-arịa ọrịa nke moto nchikota na muscle rigidity.
  • Na digestive usoro, ndị na-esonụ na-akpata: ọgbụgbọ na vomiting (adịkarịghị), afọ ntachi, afo cramps, akọrọ ọnụ, ekwe omume nke anorexia na, n'ikpeazụ, hepatotoxicity.
  • Cardio vaskụla usoro: arrhythmia, na mberede ọnụ ma ọ bụ na-abawanye na ọbara mgbali.
  • Akụkụ okuku ume na usoro: ike mgbochi nke akụkụ okuku ume center ma ọ bụ atelectasis.
  • E nwekwara ohere ndị na-esonụ nfụkasị Jeremaya: otutu, ọzịza nke ihu na akpịrị, itching, bronchospasm, laryngospasm, na urticaria.
  • N'akụkụ nke ọzọ mmetụta site n'iji codeine phosphate (na Latin, na mberede, na-ada codeinum) agụnye oké sweating, nta euphoric ala. Nakwa dị ka ihe ize ndụ nke dabeere na ogologo usoro ojiji (karịsịa buru ibu).

N'ezie, ihe ize ndụ nke n'elu kwuru banyere mmetụta bụ nnọọ obere. Ee, mgbe ịdị iche iche site edinam ime ihe.

mgbaàmà nke ovadozu

gụnyere ndị na-esonụ phenomena Mgbaàmà nke-adịghị ala ala ovadozu: uche mgbasasị, oké dizziness, nervousness na ime ihe ike, ụfụ, n'ozuzu adịghị ike nke ahụ na ọbara mgbali tụlee. Na oké ikpe, e nwere a elu puru nke ọnwụ nke nsụhọ ma ọ bụ amaghị onwe mmalite. Iri Mmadụ Ahụ ọgwụgwọ ma ọ bụ ovadozu pụrụ ịbụ nnọọ ogologo oge na-adịghị mfe. N'ọnọdụ nsi kwesịrị na-asa si afo, enwetaghị ya ume ma na-akwado obi ọrụ. Mgbe ụfọdụ, ihe ezi uche dị naloxone ogwu ogbugba, nke bụ a kpọmkwem na-eti ọkpọ nke opioid analgesics.

Special ntụziaka n'oge ọgwụgwọ

Mgbe e nwere a mgbake usoro mgbe codeine ovadozu ma ọ bụ ọgwụgwọ maka ya ahụ riri, ọrịa kwesịrị izere ịṅụ mmanya na-aba n'anya. Nke bụ eziokwu bụ na n'oge ọgwụ mmadụ dịtụ dulled na-elekwasị anya na ọsọ psychomotor Jeremaya mere. Mmanya pụrụ nanị ime ka ọnọdụ ndị siri ike. Na o nwere ike a na-adịghị mma mmetụta na a onye na arụmọrụ nke pụrụ ịdị ize ndụ-eme.

Ọ kwesịrị nlebara anya pụrụ iche n'oge ime na nwanyi. N'ezie, ojiji nke codeine nwere ike ime ka a na-egbu oge na osifikeshịọn, na mgbe ụfọdụ ozugbo nnyefe - prolongation. Ke ofụri ofụri, njakịrị na ọjọọ. N'ikpeazụ, dị ka e kwuru n'elu, na ụmụaka, ke ofụri ofụri, ekwesịghị iri codeine. Na nke a, na e nwere a bukwanu puru nke omume nke paradoxical Jeremaya mere, dị ka ụmụaka amụbawo uche mmetụta nke opioid analgesics.

legality

Na Russia, e nwere ugbu a a ụgwọ, akpan na ọgwụ ọjọọ n'ụzọ codeine. Ya mere, ịzụta ya na a na-ere ọgwụ na-enweghị a ọgwụ nwere ike ịbụ. Nso nso, na ojiji nke codeine omenala malitere ịgwa ndị ọha na eze, dị ka ewu ewu na nke ọgwụ na-eto eto exponentially. Na ọtụtụ ụzọ a "n'uru" nke American hip-iwuli elu nka onye na-na-akwado iji Purple mmanya na-egbu - a pụrụ iche ọṅụṅụ nwere elu doses nke codeine. Dị otú ahụ sirop nwere a pinkish-acha odo odo hue, gịnịkwa mere otú ahụ pụrụ iche aha. Mgbe na-aṅụ mmiri mmiri, ị ga-ezute a mmetụta nke nwayọọ anuri yiri ecstasy na opiates, nke na, n'eziokwu, na-ezo codeine. Songs of American rappers mgbe nwere ederede, na-atụ aka na Ịhazi ojiji nke Purple mmanya na-egbu. Site n'ụzọ, na Onye Okike nke a ije - Dj ịghasa. Ọ nwụrụ mgbe ọ dị afọ 29 si ịṅụfe ọgwụ ike ókè nke codeine.

Ọ kwesịkwara kwuru na codeine hụrụ ndị ọzọ ọgwụ, gụnyere ihe nile di iche iche nke fever, protivomigrenoznye na ndị ọzọ. Na nke a, ọtụtụ ọgwụ e iwu maka ire nke dị n'ókèala Russia. Ma n'ihi na iwu na-akwadoghị nkesa na ire nwere ike ịbụ na-ruo 12 mkpọrọ afọ.

Ná mmechi

Codeine nwere n'uju akporo, dị ka ya na mmetụta na-ahụ mmadụ ike. Ọ nwere ike na a pụtara mkpirikpi oge ịgbanwe uzọ nke a ọnọdụ ahụ ike nke onye ahụ. Kacha nkịtị ụdị codeine (phosphate) - a ntụ ntụ nke bụ ngwa ngwa soluble n'ime mmiri. N'ihi ya Njirimara, ọ e ọtụtụ-eji nkà mmụta ọgwụ. Otú ọ dị, dị ka a na-ahụkarị na opiates, umi seeped ngwa ngwa banyere n'okporo ámá, nke nwere a ezighị ezi mmetụta na ndị mmadụ na-ewe ya, ndị na-esi nke bụ nke nwere ike igbu.

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