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"Excedrin": ogbo. Ọgwụgwọ maka migraine "Excedrin": reviews, ahịa, analogs

Migraine - nke a bụ ọrịa, nke ike-agafere enweghị analgesics. The agha bụ ike-adịgide adịgide maka 4 ụbọchị. The nwoke na oge a na-efunari ya ike na-arụ ọrụ. N'otu oge ahụ ọ na-eji ike na nkà mmụta ọgwụ tufuo nke throbbing mgbu. Ma, dị mwute ikwu na ọtụtụ n'ime ngwá ọrụ ndị na ike iwepụ dị otú ahụ erughị ala, na-eri ahụ na-eduga eziokwu ahụ bụ na ọrịa na-aghọ ala ala. Modern pharmacology azụlitewo a oké ọgwụ ọhụrụ. N'aka, ọma tufuo migraine, na-ebelata ikike o nwere ịrụ ọrụ, ma ọ bụghị na-eri ahụ, ọgwụ bụ "Excedrin". Analogs nke ọgwụ abụghị obere irè.

nkenke nkọwa

Ọgwụgwọ maka migraine "Excedrin" bụ a jikọtara nkwadebe nke ìgwè nke analgesics-antipyretics. Ọ na-eji maka oké isi ọwụwa. Ọma pụtara "Excedrin" si oké isi ọwụwa. Na nke a, ọ pụrụ ọbụna gbochie agha.

The mejupụtara nke ọgwụ

The ọgwụ na-irè dị na ya Efrata. The na nkà mmụta ọgwụ nwere:

  • acetylsalicylic acid;
  • caffeine;
  • paracetamol.

Ọ bụ ekele ndị a ọcha nwere iche iche mmetụta na ahu. N'ihi ya, na-ekwe nkwa ozugbo mmetụta, n'ụzọ zuru ezu kwụsịrị n'ọdụ ụgbọ mmiri mgbu.

Paracetamol ke ichekwa 250 mg, Acetylsalicylic acid - 250 mg, na caffeine - 65 mg otu mbadamba e tinyere ọgwụ ọjọọ "Excedrin". The mejupụtara otú n'ime ebe a pụtara n'ọrụ Efrata dị nnọọ ịrịba ama. Ọ bụ ya mere na-atụ aro iji ọgwụ ọjọọ na oké ịkpachara anya. Ọrịa ga-gaa na akaụntụ na onunu ogwu na gafere ya.

Ke adianade do, a ọgwụ na-agụnye inyeaka Efrata:

  • giproloza;
  • microcrystalline cellulose;
  • stearic acid.

Mmetụta na-ahụ

Mbadamba migraine "Excedrin" mere nke atọ dị iche iche ihe nke nwere dị iche iche Njirimara. Ha Nchikota na-enye ohere ka tufuo ihe mgbu nke ọ bụla okike. Ebe ọ bụ na migraine ọgụ esonyere a zuru ezu ogologo na oké ahụ erughị ala, ka tufuo ya ga-nnọọ ike na nkà mmụta ọgwụ. Na ndị dị otú bụ ọgwụ "Excedrin".

Gịnị ngwá ọrụ a nwekwara owụt ya mmetụta na nso utịp? Azịza nke ajụjụ dabeere na mmetụta na ozu nke ọ bụla akụrụngwa dị na ọgwụ:

  1. Paracetamol. The umi nwere a elu mgbochi mkpali na antipyretic Njirimara. Ọ bụ ike na-emetụta ụbụrụ center na bụ maka ịchịkwa okpomọkụ na hypothalamus. Ọrụ dị mkpa mkpochapu migraine ya nwere mgbochi mkpali quality, n'ihi na ahụ ọkụ na-abụghị nke na mgbaàmà nke ọrịa.
  2. Acetylsalicylic acid. Akụrụngwa dị iche akpọ antipyretic Njirimara. Ọ bụ ike ịkụda na iwepụ mbufụt. Na nke a na-ebelata ihe mgbu. Acetylsalicylic acid pụrụ igbochi omume egbochi mkpụkọ nke ọbara. Ọ na-akwụsị na usoro nke ha n'usoro na na cellular larịị, n'ụzọ zuru okè enhances ọbara na-nanị ire ọkụ ebe.
  3. Caffeine. The ọrụ nke a umi iji belata ihe mgbu kasị dị ịrịba ama. Ịṅụ Ọgwụ Aspirin na paracetamol nwere ike nwa oge kpochapụ ahụ ala. Caffeine nwere mmetụta dị mma n'ebe ọbara na ụbụrụ na-enyere aka bibie ndị na-akpata ọrịa. Ọzọkwa, ọ na-akpali iku ume ma na vasomotor emmepe, na-akwalite mgbasa nke narrowed ọbara arịa, na-egbochi platelet nkịtị. Caffeine bụ magburu onwe Aka ike ọgwụgwụ na-ehi ụra. Ọ budata enwekwu ndị arụmọrụ nke organism na ya ụda, otua kwalite onye ọrịa ahụ n'ozuzu ike. The Nchikota aspirin na umi ike ime ọbara eruba na ghaghị emetụta ụbụrụ arịa.

Pathologies nke nkwadebe na-etinyere

Ọ bụ amamihe na-eji "Excedrin" ọgwụ n'ihi ihe mgbu ọrịamkpokọta nke dịkwa nwayọọ na agafeghị oke osisi ike nke dị iche iche si malite:

  • migraine;
  • isi ọwụwa;
  • neuralgia;
  • eze mgbu;
  • myalgia, arthralgia (erughị ala na nkwonkwo na akwara);
  • algomenorrhea (mgbu mgbe nanso);
  • feverish syndrome.

Pharmacokinetics

N'ọnọdụ ka ukwuu, ahụ na nkà mmụta ọgwụ "Excedrin" ezi uche ọma anabata. Consumer reviews n'ụzọ zuru ezu gosi na nke a. Mmetụta dị otú ahụ nke ọgwụ a chọrọ nke ya mmiri:

  1. Paracetamol n'ụzọ zuru okè etinye obi gị dum na eriri afọ tract. Ọ na-metabolized na imeju, akụrụ na-anyụpụ ka glucuronide na sulfate conjugates. Na-erughị 5% nke ihe onwunwe exits na unmodified ụdị. Ebe ọ bụ na plasma protein nkekọ bụ ntakịrị mgbe eji a ot ọgwụgwọ dose. Ma na na-abawanye na nke ikpeazụ - na-amụba. Hydroxylated metabolite guzobere obere na imeju n'okpuru nduzi nke mbuaha oxidases na-emekarị na-neutralized site na nkịtị na glutathione, nwere ike akpọkọtara na ịṅụfe ọgwụ ike ókè nke paracetamol na ime ka imeju mebiri.
  2. Acetylsalicylic acid kpamkpam na ngwa ngwa etinye obi gị dum. Ọ na-hydrolyzed na digestive tract, ọbara na imeju. N'ụdị a salicylates. Ọzọkwa, ha na-metabolized na imeju.
  3. Caffeine na-ngwa ngwa etinye obi gị dum n'ụzọ zuru ezu. The kacha ịta na ahụ a hụrụ maka 5-90 nkeji mgbe ojiji nke ego na ihe efu afo. Excretion emee ka a n'ihi nke hepatic metabolism. The umi a na-ekesa ihe nile mmiri ahụ. Communication na plasma protein bụ 35%. Akụrụngwa kpamkpam metabolized na anyụpụ site na akụrụ ya.

dosing Usoro

Adabara onu ochichi pụtara "Excedrin". The na nkà mmụta ọgwụ na-eji n'oge ma ọ bụ mgbe a nri. Ọ na-atụ aro na-aṅụ mmiri na nnukwu quantities.

Single dose n'ihi na ndị okenye na-eto eto (site na afọ 15) - 1 mbadamba ọ bụla 4-6 awa. Ọ bụrụ na mmadụ na-ele ihe ịrịba ama nke na-abịanụ migraine, ọ na-atụ aro iji otu mgbe 2 ọgwụ. Nke a ga-egbochi ihe agha nke ọrịa. Otú ọ dị, onye kwesịrị icheta na-eri karịa 6 nkeji kwa ụbọchị na-nditịm ajuru aju.

mkpa ịdọ aka ná ntị

Irè na nkà mmụta ọgwụ na-ekwe na-etinye maka egbu mgbu erughị ala ruo ụbọchị 3. N'oge a, onye ọrịa kwesịrị ịkpọ na dọkịta gị, onye ga-họrọ zuru okè ọzọ ụzọ nke na-alụ ọgụ ka ọrịa.

Mgbe ụfọdụ, ọrịa na-atụ aro ịgbatị na ojiji nke ọgwụ. Ma mkpebi dị otú ahụ nwere ike na-adabere na nke kwesịrị ekwesị na-egosi na a ọkachamara. Rie mkpụrụ ọgwụ migraine "Excedrin" nwere ihe karịrị 3 ụbọchị adịghị atụ aro. Amụba dose ike nke na-eme ka oké njọ pụta. Dị ka imeju mmebi ruru ka ìgwè metabolites ke idem.

mmetụta

The iji ọgwụ ike n'ezie nwere nti utịp ke idem. Ebe ọ bụ na o nwere ọtụtụ mmetụta pụtara "Excedrin". Drug analogues nwere ike ikwu n'imeso dọkịta, ma ọ bụrụ na n'elu-e kwuru ọgwụ na-adịghị ruru eru ka onye ọrịa.

Ya mere, ndị na-esonụ mmetụta:

  • ọgbụgbọ, vomiting;
  • gastralgia;
  • hepatotoxicity;
  • erosive na ọnyá eriri afọ ọnya;
  • nephrotoxicity;
  • nfụkasị Jeremaya;
  • amụba mgbali;
  • tachycardia;
  • dizziness;
  • bronchospasm;
  • isi ọwụwa;
  • bịara ikiri ọhụụ;
  • ibelata na platelet aggregation ;
  • tinnitus;
  • hemorrhagic syndrome (ọbara ọgbụgba goms, epistaxis, purpura);
  • ịza aza exudative erythema (ma ọ bụ Stevens-Johnson syndrome);
  • ntị ochichi;
  • na-egbu egbu epidermal necrolysis (ma ọ bụ Lyell si syndrome);
  • akụrụ ọrịa (Chance papillary necrosis);
  • mmepe na ụmụ Raynaud si syndrome (hyperpyrexia, metabolic acidosis, ọrịa nke ụjọ usoro na psyche, vomiting, ndiiche imeju ọrụ).

Contraindications anata

N'ụzọ dị mwute, ọgwụ agaghị irè maka mmadụ nile. Mgbe n'aka nwere ọtụtụ contraindications. Ha na-n'aka-sonye na akaụntụ tupu n'itinye. Ma obi nkoropụ ma ọ bụrụ na ndị nkà mmụta ọgwụ adịghị abịa enweghị akwụ ụgwọ. The ịga dibịa bụ nnọọ mfe iji dochie ngwá ọrụ "Excedrin". Analogs ekwe iji nweta na-anara nke N'ihi.

Ọgwụ na-contraindicated na-eso pathologies na ọnọdụ:

  • Hypersensitivity ka Efrata;
  • eriri afọ ọnyá na nnukwu ogbo;
  • bronchial ụkwara ume ọkụ,
  • agba ọbara eriri afọ;
  • ntighari dịghị òkè polyposis (paranasal sinuses);
  • ekweghị ibe nọrọ na NSAIDs;
  • usoro ịwa ahụ na-eso ọbara na-agba;
  • hemorrhagic diathesis;
  • ọbara mgbali;
  • hemophilia;
  • gipoprotrombinemii;
  • portal ọbara mgbali;
  • glaucoma;
  • oké ischemia nke obi;
  • beriberi K;
  • enweghị glucose-6-phosphate dehydrogenase;
  • gbasara akụrụ odida;
  • ime;
  • lactation;
  • nsogbu ihi ụra;
  • ogwe;
  • Ụmụaka afọ (a ọgwụ na-adịghị emetụta afọ 15).

ovadozu nke na nkà mmụta ọgwụ

Medicine "Excedrin" migraine kwesịrị na weere na doses gosiri n'elu. Ebe ọ bụ na mmetọ gị n'ụlọnga nwere ike ime ka a ìgwè wetara ihe mgbaàmà.

About ovadozu nke paracetamol egosi ndị na-esonụ atụmatụ:

  1. N'oge n'ụbọchị mbụ e icha mmirimmiri anụ ahụ, vomiting, ọgbụgbọ, abdominal mgbu, mkpọchị glucose metabolism, anorexia, metabolic acidosis.
  2. Mgbe 12-48 awa nke ime ihe kwere omume ihe ịrịba ama nke imeju odida kwuru na progression nke encephalopathy. N'ihi na oké ovadozu ekwe omume - atụbọ ma nwụọ. E nwere ike gbasara akụrụ odida, Bilie tubular necrosis, pancreatitis, arrhythmia.

Ovadozu iwe na acetylsalicylic acid, nwere ndị na-esonụ mgbaàmà:

  1. Nwayọọ - vomiting, ọgbụgbọ, dizziness, bịara ikiri ọhụụ, tinnitus, isi ọwụwa.
  2. Na oké nsi - mkpụmkpụ nke ume, cyanosis, dyspnea, nnyapade oyi ajirija, akụkụ okuku ume na acidosis, akụkụ okuku ume na mkpọnwụ.

Abuse mere site caffeine na-kwupụtara na-esonụ mgbaàmà:

  • gastralgia;
  • n'ahụhụ, nchegbu;
  • mgbagwoju anya;
  • erughị ala;
  • akpịrị ịkpọ nkụ;
  • arrhythmia;
  • Ugboro urination;
  • tachycardia;
  • hyperthermia;
  • ihe mgbu ka ukwuu na uche;
  • tremor;
  • ịkụ na nti;
  • ọgbụgbọ, vomiting (mgbe ụfọdụ na ọnụnọ nke ọbara);
  • akwụkwụ ọdịdọ.

Ọ bụrụ na ovadozu kwesịrị ịchọ ahụike mberede enyemaka. N'oge mbụ 4 awa ọ na-atụ aro na-asa na afo, eji vomiting. Laxatives ga-iwesa na pụtara "ọrụ carbon".

analogues na nkà mmụta ọgwụ

Cheta na ọ bụla ọgwụ ga-kenyere onye dọkịta, ebe onye ọ bụla gị n'ụlọnga nwere ya na-egosi na contraindications.

Na naanị a dọkịta bụ ike ịnọchi anya ọzọ ọgwụ na nkà mmụta ọgwụ "Excedrin". Analogs nke ugbu a akụrụngwa dị ka ndị a:

  • "Akvatsitramon".
  • "Atsifein".
  • "Askofen".
  • "Kofitsil plus."
  • "Tsitramarin".
  • "Migrenol Extra."
  • "Tsitramon".
  • "Tsitrapar".

The na-eri nke ọgwụ

N'ihi na ihe niile ya arụmọrụ, ọnụ ọgwụ na-akwụ ụgwọ na-eji ọkụ "Excedrin" si oké isi ọwụwa. Price nke ngwugwu (10 mbadamba) dịgasị na nso nke 120-150 rubles. The na-eri nke nkwadebe nke 20 ọgwụ nke 210-250 rubles.

Mmekọrịta ndị ọzọ ọgwụ ọjọọ eme ihe

Ọrịa na-eji ọgwụ ọjọọ, "Excedrin" ga-aghọta na o nwere ike welie utịp ke idem ọzọ n'aka dị ka:

  • "Heparin";
  • anọ anticoagulants;
  • "Reserpine";
  • hypoglycemic ọgwụ ọjọọ;
  • steroid homonụ.

Rịba ama na nke imekotaotuugbo ojiji nke ego "Excedrin" na ndị ọzọ NSAIDs nwere ike ime ka mmetụta. Ka ihe atụ, mmekọrịta protivopodagricakih ọgwụ ọjọọ, antihypertensive ọgwụ ọjọọ, pụtara "Furosemide" na-eduga ná ala arụmọrụ nke ndị a dị iche iche nke ọgwụ ọjọọ.

n'ji uche

Ọ bụla ọgwụ nwere (sokwa na-agwọ "Excedrin") Ibọrọ, ma nke oma ma na-ezighị ezi.

Ụfọdụ na-eji ọkụ gwa hoo haa na, ọ gbalịrị ọgwụ ozugbo, agaghị akụkụ na ha. Ọtụtụ ụmụ nwaanyị bụ ngwá ọrụ dị irè na ya obere akpa. Ị dịghị mara mgbe mgbu agha ga chụkwute gị. Ndị dị otú ahụ ọrịa na-achọpụta na otu mbadamba ike hour kpochapụ wetara ihe mgbaàmà. Na na ikpe nke oké oké isi ọwụwa eliminates mgbu ọgwụ ọgwụ 2 "Excedrin". Ibọrọ na-egosi na ndị magburu onwe arụmọrụ nke ngwá ọrụ.

Ndị ọzọ na-eji ọkụ jide a dị iche iche echiche, na-ezisa abaghị n'ihe nke ọgwụ. Ha na-ekwu na-arụ ọrụ bekee ọgwụ nwere ike zụrụ n'otu n'otu bụ ihe dị ọnụ ala karịa ahịa ọgwụ. Otú ọ dị, ndị a ahịa na-echefu na ịdị irè ọgwụ dị ka a n'ihi nke nri Nchikota niile mmiri na zuo ezu onye ọ bụla ọzọ n'ụzọ zuru okè.

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