Ahụ ikePreparations

Metoprolol-ratiopharm

Metoprolol-ratiopharm esịne ke otu ọgwụ ọjọọ na-eji na ọgwụgwọ nke ọrịa obi. Ọgwụ bụ nke pharmacological ìgwè nke beta-blockers.

Metoprolol mbadamba nwere hypotensive, antiangialnym na antiarrhythmic mmetụta. The ọgwụ na-egbochi mmepe nke migraine.

Dị ka nhọrọ beta blocker, metoprolol-ratiopharm mgbe eji ọgwụgwọ doses ajụ nwere ntakiri mmetụta na akụkụ na-ebu beta-2-adrenoceptors (skeletal muscle, pancreas, elu ọbara ezigbo uru nke akpanwa, na bronchi), na na-na carbohydrate metabolism. N'ihi ya atherogenic edinam owụt ke ukem udomo dị ka mgbe iji propranolol. Mgbe e ke nnukwu doses Metoprolol-ratiopharm na-akpa a igbochi utịp ke beta-1 na beta-2 andrenoretseptory.

N'itinye n'ime akara zuru absorption (95%). Metoprolol-ratiopharm ngwa ngwa na-ekesa na anụ ahụ, penetrates site na placental mgbochi, BBB.

The ọgwụ na-metabolized na imeju, na metabolites adịghị eme ka a pụrụ iche onyinye ọrụ nke beta-adrenoceptor igbochi agwa.

The ọgwụ na-owụt maka ọbara mgbali (ma onwe ha na dị ka akụkụ nke Nchikota ọgwụ na ndị ọzọ antihypertensive ọgwụ), n'ihi na obi anaghị ekwe ọtọ ọdịdị esonyere tachycardia. Kenye metoprolol na ischemic ọrịa obi: myocardial infarction (dị ka a abụọ mgbochi), rịaworo (dị ka ọdịdọ mgbochi). Ọgwụ gosiri maka mgbochi nke ventricular arrhythmias na supraventricular tachycardia, nakwa dị ka migraine.

The agwọ ọrịa eji na-ekwesịghị na ọrịa na-arịa ọrịa shuga mellitus, ụkwara ume ọkụ, metabolic acidosis na gbasara akụrụ (imeju) ọdịda, thyrotoxicosis, myasthenia gravis, psoriasis, occlusive elu vaskụla ọrịa, afọ ime, na nká.

Metoprolol-ratiopharm. ntụziaka

Mbụ onunu ogwu na ọbara mgbali bụ 50 mg. Bụrụ na nke ezughi oke ọgwụgwọ mmetụta, ọ nwere ike na-amụba ka 100-200 mg ma ọ bụ n'ihu nzube ọzọ antihypertensive ọgwụ ọjọọ. Daily dose (kacha) bụ 200 mg.

Ọgwụ e ji ọnụ na, na mmiri, otu ugboro n'ụbọchị ozugbo a nri. Mbadamba ekwesịghị ata ata.

Dị ka mgbochi maka mgbochi nke rịaworo ọgụ mbụ kwa onunu ogwu nke ọgwụ nke 50 mg. Bụrụ na nke ezughi oke irè nke ọgwụgwọ ọ nwere ike na-amụba ka 100-200 mg ma ọ bụ yana ọrụ antiangialnyh ọzọ ọgwụ. Oke onunu ogwu kwa ụbọchị - 200 mg.

Iji gbochie migraine ọgụ aṅụ ọgwụ kwa ụbọchị nke 100-200 mg.

Site 50 ruo 200 mg nke ọgwụ ndinọ na ọtọ gbasara obi ọrịa so site tachycardia.

Mgbe mgbochi (nke abụọ) myocardial infarction agwọ ọrịa na-ndinọ na a onunu ogwu nke 200 mg kwa ụbọchị.

Na gbasara akụrụ insufficiency, na onunu ogwu adịghị achọ mgbazi. Dabere na-adakarị ọnọdụ hepatic ọdịda nwere ike ime ndị dị otú ahụ a mkpa.

Na-ewere ọgwụ na-Ugboro oghom ihe dị ka bradycardia, a oyi snap ke ala na nsọtụ, orthostatic hypotension (gụnyere na syncope), ike ọgwụgwụ, ajụ obubu, nchegbu, mụbara ụjọ ogwe, mmekọahụ dysfunction, ọgbụgbọ, abdominal mgbu, afọ ọsịsa ma ọ bụ afọ ntachi, dyspnea na mgbalị siri ike.

Kagbuo ọgwụ emepụta nwayọọ nwayọọ mgbe mbenata onunu ogwu maka izu abụọ. Ọ ga-kwuru na nkọ ojuju nke ego nwere ike ịkpalite ụba ọbara mgbali, n'ihe ize ndụ nke rịaworo ọgụ.

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