Ahụ ike, Preparations
"Antabuse" mkpụrụ ọgwụ. Nyocha, price ndu
Ọ na-akpọ aṅụrụma a ọrịa na e ji ihe riri ka ethanol na ahụ na uche na nduzi na ya. Nke a na ụdị nke mmegbu. Na steeti a, ọnwụ nke na-achịkwa ego mmanya na-egbu mmanya enwekwu ndidi ya (iji nweta afọ ojuju mmanya mgbe niile na-amụba dose) na ndọrọ syndrome etịbe, na-emetụta akụkụ ahụ ndị na-egosi na ebe nchekwa gafee.
Ọrịa na-arịa aṅụrụma, na-akpọ ndị aṅụrụma. Na-emeso ndị ọrịa kwesịrị uche na ọkpụkpụ. Ọtụtụ mgbe, ndị dọkịta ji nye iwu ka a ọgwụ ndị "na Antabuse". Ntuziaka maka ojiji, price nke ọgwụ, ọgwụ na reviews na-egosi n'okpuru.
Mbukota, udi, na Ọdịdị nkọwa
Na ihe na-etolite ọgwụ a na-eresị "Antabuse"? Nleba na-akọ na ndị dị otú ahụ a usọbọ nwere ike zụrụ n'ụdị ọcha, gburugburu effervescent mbadamba. Ha na-ewepụghị, beveled onu, ize ndụ ma na-akara «CD» na «C» na-abụghị n'akụkụ nke ize ndụ.
The mejupụtara nke a ọgwụ na-agụnye disulfiram. E wezụga ya, nkwadebe nwere ọka starch, povidone, sodium hydrogencarbonate, tartaric acid, colloidal sịlịkọn dioxide, talc, microcrystalline cellulose na magnesium stearate.
Mbadamba "Antabuse" enịm ke plastic containers na ngwugwu katọn.
pharmacodynamic e ji mara
Gịnị bụ ọgwụ "Antabuse"? Manual na-ekwu na nke a pụtara antialcoholic. Ọ na-egbochi acetaldehyde dehydrogenase, nke a na-metabolism nke ethanol. Oge ya ọxịdashọn usoro na-eme ka ìgwè mmanya na mmepe nke siri ike igbu egbu, sochiri arọ mmetụta dị ka a throbbing mgbu na mkpọtụ na isi, tachycardia, palpitation, Mbelata ke ọbara mgbali, ọgbụgbọ, bịara ikiri ọhụụ na vomiting.
Dị ka ndị ọkachamara, ndị a wetara ihe mgbaàmà na-eme ka mmepe nke haziri mpiaji mkporomaasi ka mmanya.
pharmacokinetic Njirimara
Olee otú ndị absorption nke "Antabuse" ọgwụ ọjọọ? Manual na-egosi na ọgwụ a na-etinye obi gị dum site na 70-80%. Ọ bụ ukwuu soluble na lipids na nēche imubanye na abụba na-ebusa.
N'ọrụ umi nke gị n'ụlọnga na-nnọọ ngwa ngwa metabolized, n'ihi na gbanwee metabolite - methyl Ester dietiltiokarbaminovoy acid. Ya elu ọbara kasịnụ kpebisiri ike mgbe 4 h. Ọ bụ ezie na ọrụ na mmekọrita acetaldehyde dehydrogenase a hụrụ nanị mgbe ụbọchị atọ.
The ọkara ndụ nke ọgwụ bụ 10 awa. Ọzọkwa, ya ọrụ megide aldehyde dehydrogenase nọgidekwara ogologo. Ya mere, mgbe a kagbuo mmetụta nke mbadamba na-hụrụ maka a n'ihu 7-14 ụbọchị.
The ọgwụ na-egosi na mmamịrị, na emezughị site eriri afọ na exhaled ikuku.
na-agba akaebe
Mgbe ụfọdụ, ndị kasị dị irè iji ọgwụ na-akpa àgwà "Antabuse"? Nyocha kọrọ na a owuwu na ọtụtụ-eji maka mgbochi nke nlọghachi azụ na ọgwụgwọ nke na-aba n'anya na nduzi na aṅụrụma.
contraindications
Mgbe ị na-ekwesịghị iri "Antabuse" mbadamba? Ọbịa ọkachamara na-ekwu na-ewere ọgwụ na-ekwesịghị kenyere ma ọ bụrụ na:
- glaucoma;
- neuritis nke optic na auditory akwara;
- akpa ume ụkwara nta;
- obi na vaskụla ọrịa na (e.g., post-infarction ekwu, kwupụtara cardiosclerosis, atherosclerosis nke ụbụrụ arịa, hypertensive ọrịa, aortic aneurysm);
- polyneuritis nke ọ bụla si;
- arịa ọrịa shuga;
- emphysema, bronchial ụkwara ume ọkụ;
- thyrotoxicosis;
- iche echiche ọrịa, Akwụkwụ na-adọ na epileptiform syndrome;
- ịza aza akpụ;
- oké hepatic na gbasara akụrụ odida;
- ọrịa nke hematopoiesis;
- exacerbation nke peptic ọnyá afọ ọrịa;
- ime;
- hypersensitivity.
Ọzọkwa mara na nke a ọgwụ bụ ikwu contraindications:
- afọ 60 afọ;
- mmetụta nke a ọrịa strok na mmapụta mgbaàmà;
- peptic ọnyá afọ (gụnyere na ngbaghara);
- precipitates a psychosis.
Drug "Antabuse": ntuziaka maka ojiji
Anti-mmanya Erere price depụtara na njedebe nke isiokwu. Ga-ha n'ime ½ mbụ etisasịwo ke otu iko mmiri.
A, dọkịta nye iwu 200-500 mg nke ọgwụ ozugbo ma ọ bụ ugboro abụọ n'ụbọchị. Mgbe 7 ụbọchị, ijide n'aka na-eji disulfiram-mmanya ule. Ke ukem na n'ikuku nke 500 mg nke agwọ ọrịa ndidi ọṅụṅụ 20-30 ml nke vodka. Ọ bụrụ na mmeghachi omume na-adịghị ike, mgbe ahụ, dịkwuo dose mmanya 20 ml.
Nke a ule na-ugboro ugboro ugboro ugboro. Mgbe e mesịrị ballroom kenyere mmezi onunu ogwu nke 200 mg kwa ụbọchị maka 1-3 afọ.
oghom Jeremaya mere
Mbadamba "Antabuse", nke ratings-ọkọnọ n'okpuru nwere ike ime ka ndị na-esonụ mmetụta:
- ịba ọcha n'anya, asthenia, metal uto ke inua;
- cutaneous ngosipụta, polyneuritis ụkwụ;
- ebe nchekwa ọnwụ, ụbụrụ ọzịza, isi ọwụwa;
- myocardial infarction, gbasara obi arrhythmias;
- akụkụ okuku ume na ọdịda, obi ida;
- optic neuritis, ọrịa ụbụrụ thrombosis arịa;
- psychoses, rịaworo.
Agwọ ọrịa "Antabuse": reviews nke dọkịta na price
The na-eri nke mgbochi mmanya mbadamba bụ banyere 450-600 rubles (dabere na dose na ego kwa mkpọ).
Dọkịta na ndị nye iwu ndị dị otú ahụ a ọgwụ, ozugbo dọrọ aka ná ntị nke oké njọ nsogbu na nwere ike ime na a ọrịa na ndabere ọ ga-ewe. Ya mere machibidoro kpam kpam na-emeso onwe gị ma ọ bụ a ezo site na ndidi.
Ọ kwesịkwara kwuru na ọtụtụ ndị ọkachamara na-ekweta na irè ọgwụ ọjọọ na-ebelata agụụ maka mmanya, ọ dịghị. Na usoro a bụ bụghị ọgwụ. Ọ nanị na-akwalite a ufọk ufene kwụsịtụkwara.
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