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"Lopedium" Mbadamba: ntụziaka ntuziaka, reviews

"Lopedium" - a ọgwụ mwute peristalsis. Bụ a gelatin Capsule na a ike shei, na-ese na agba ntụ ma ọ bụ ọchịchịrị akwụkwọ ndụ akwụkwọ ndụ na agba (na ha nwere a whitish homogeneous ntụ ntụ) ma ọ bụ na-acha ọcha mbadamba.

pharmacological Njirimara

Mbadamba "Lopedium" (ntuziaka maka ojiji n'isiokwu a) na-ekewet nke a umi ike nke na kọntaktị na nsia opiate anabata. Site na nke a na njikọ ya gbochie ntọhapụ nke acetylcholine na prostaglandin. N'ụzọ dị otú a a usu-ebelata nke ukwu enwekwu peristalsis na-adịru nwa ọdịiche Itie nri site na digestive tract. Ọzọkwa nsia mgbidi banye ọzọ oke mmiri-abịa na ụda olu nke sphincter uru.

Pharmacokinetics

Ọtụtụ n'ime loperamide, banyere n'ime ahu na-etinye obi gị dum na eriri afọ ya, Otú ọ dị, n'ihi na kpụ ọkụ n'ọnụ akpa-ngafe metabolism, systemic bioavailable bụ naanị a nkeji iri na ise nke a percent.

Site research ya na a hụrụ na a ọgwụ a na-ekesa na-akwanyere ndị nsia mgbidi, ma si otú na-ejikọ na-anabata longitudinal muscular uwe oyi akwa. Ukwuu n'ime loperamide ejikọ na-edozi ahụ, karịsịa albumin.

Mbadamba "Lopedium" (ntụziaka ntuziaka classifies ha dị ka mma ọgwụ ọjọọ) fọrọ nke nta kpamkpam etinye obi gị dum site na imeju, ebe ha na-metabolized, conjugated na anyụpụ na bile. N'ihi na oké ufiop mmetụta nke mbụ Itie site imeju nkwadebe, ịta nke ọgwụ na ọbara na-budata belata, mgbe fọdụrụ nnọọ ala. The ọgwụ na-kpamkpam anyụpụ site iri na otu - iri na anọ awa.

egosi

"Lopedium" (mbadamba) ntụziaka ntuziaka na-atụ aro na na ikpe nke na-adịghị ala na nnukwu afọ ọsịsa. A ọgwụ ike ga-ndinọ ka ndị mmadụ aka na njem ( "njem nleta afọ ọsịsa"). Na nke a, ọgwụgwọ kwesịrị ụbọchị abụọ. Otú ọ dị, n'ihe banyere nchọpụta nke ọbara na stool dịghị mkpa ka na-eji nkà mmụta ọgwụ na-ekpebi ihe na-akpata ọrịa na dọkịta.

contraindications

Unu na-eji mbadamba nkume na ihe omume na e nwere hypersensitivity ka loperamide hydrochloride ma ọ bụ ka ọ bụla ọzọ mmiri nke nkwadebe.

Isi contraindications maka ọrịa:

- nje enterocolitis, n'ihi omume nke ụfọdụ microorganisms:

- nnukwu ọnyụnyụ ọbara, Bilie ọbara afọ ọsịsa nakwa fever.

Na ijikọta ọgwụ ọ bụla ọgwụ nje mkpa na oké ịkpachara anya. Jide n'aka na-agwa dọkịta gị.

Unu na-eji mbadamba nkume "Lopedium" (ntụziaka ntuziaka adọ aka ná ntị ọrịa) na mmepe nke afọ ntachi, bloating ma ọ bụ nsia mgbochi. Zere ego ma ọ bụrụ na ọ dị mkpa izere mmegbu nke peristalsis.

Olee otú ga-ewere "Lopedium" mbadamba

The ọgwụ ike ga-eji na ndị okenye na ụmụaka okenye karịa afọ isii. Capsule (mbadamba) ga-elo dum na a obere mmiri dị ọcha.

Na-adịghị ala ala na nnukwu afọ ọsịsa dose n'ihi na ndị okenye bụ n'etiti 4 mg Nwa (abụọ PC.). Maka ụmụaka bụ ezuru otu. The ọgwụ kwesịrị iwere mgbe ọ bụla rụrụ stool. Oke kwa ụbọchị ọnụego ụmụaka na ndị okenye bụ isii asatọ mbadamba.

Ọ bụrụ na nnukwu afọ ọsịsa mgbaàmà akwụsị n'ime iri anọ na asatọ awa, ọgwụ ga-akwụsị.

Agadi ọrịa adịghị mkpa pụrụ iche onunu ogwu ukpụhọde ndu. Otu na-aga n'ihi na ndị mmadụ na-ata ahụhụ si na ọrịa nke na akụrụ ya. "Lopedium" (mbadamba) ntụziaka ntuziaka adịghị atụ aro ka na-enye ụmụ afọ 3.

Atụmatụ nke ngwa

N'ozuzu, usoro ọgwụgwọ nke afọ ọsịsa bụ Ịhazi. Ọ bụrụ na onye ọrịa nwere ohere kọwaa etymology nke ọrịa, na nke a ọ dị mkpa iji mepụta ụdị ọgwụgwọ. Ọ bụ omume na ọgwụ kenyere ndị dibịa n'oge ngwa nke ọgwụ nje ọgwụ. Ke ukem na n'ikuku pụtara "Lopedium" (mbadamba) ntuziaka maka ojiji nke ụmụaka na-atụ aro nnọchi ọgwụ idochi electrolytes na oke mmiri. Nke a ga-eme na ihe omume na e nwere ihe ahaghị nhata nke electrolytes na akpịrị ịkpọ nkụ.

Ọrịa ndị a chọpụtara na ha nwetara immunodeficiency syndrome (AIDS), afọ ọsịsa kwesịrị ozugbo kwụsị ịṅụ "Lopedium" na ikpe nke na bloating.

"Lopedium" (mbadamba): Ntụziaka maka iji n'oge ime na ara

Dọkịta adịghị ike ikwu na-ewere ọgwụ maka ime na lactating inyom. Nke a bụ n'ihi na eziokwu na obere loperamide nwere ike ịpụta na mmiri ara. Ọ bụ ya mere ụmụ nwaanyị "na steeti" mgbe niile kwesịrị ịkpọ onye dọkịta tupu ịzụrụ na ọgwụ.

Mmekọrịta ndị ọzọ ọgwụ ọjọọ eme ihe

Ọkà mmụta sayensị na-ikpe mmekọrịta ọgwụ ọjọọ nke nwere yiri pharmacological e ji mara. Ọgwụ nwere depressant mmetụta na Central ụjọ usoro, ike ga-achọkwa na "Lopedium".

Ọ bụ uru na-arịba ama na loperamide - bụ a mkpụrụ nke P-glycoprotein. Imekotaotuugbo ojiji 'Lopedium "na quinidine na ritonavir ike ịkpata a ịrịba abawanye na ọbara ịta nke ọgwụ. The dose nwere ike mụbara abụọ ma ọ bụ ugboro atọ. A mmetụta yiri chọpụtara mgbe itraconazole na ketaconazole.

Ọ na a hụrụ na ọgwụ ọjọọ na-enwe yiri pharmacological Njirimara nwere ike welie edinam nke loperamide ọtụtụ ugboro. Ma ọgwụ ọjọọ eme ihe na-adị n'elu usoro nke na-agafe na ọdịnaya nke eriri afọ tract, na Kama nke ahụ, belata ya irè.

ovadozu

Mbadamba "Lopedium" (ntụziaka maka ojiji na-akọwa ihe mgbaàmà nke ihe ovadozu) pụrụ iduga a ọnwụ nke nchikota, isi ọwụwa, somnolence, stupor, na urinary njigide. Ọ bụrụ na ị hụrụ ihe mgbaàmà ndị yiri, ị pụrụ "Naloxone". Na obere okwu, afo-na-asa na ihe ọṅụṅụ ọrụ unyi.

oghom Jeremaya mere

Na akpụkpọ ọkụ ọkụ nwere ike kpụrụ, gụnyere Stevenson-Johnson syndrome; erythema multiforme; ozizi; itching na aṅụ.

The ọgwụ nwere ike imetụta na ụjọ usoro. Ọrịa nwere ike iro ụra, ọnwụ nke nchikota, ọnwụ nke nsụhọ, ọbara mgbali elu, na tremor.

Si digestive usoro, ọrịa nwere ike na-achọpụta a akọrọ ọnụ, afọ ntachi, ọgbụgbọ, flatulence, vomiting, ileus. Ọtụtụ ndị ọrịa nwere ike ọgwụgwụ.

Ihe ókè ịkpachara anya ga-eji ọgwụ ọjọọ ndị ọkwọ ụgbọala na-eji ígwè ọrụ, dị ka ọgwụ nwere ike ime ka iro ụra.

Hapụ ụdị, mejupụtara na mbukota

Onye ọ bụla Capsule (mbadamba) dere abụọ milligrams nke loperamide hydrochloride. E wezụga isi ọgwụ, na nkwadebe nwere inyeaka, ya bụ, talc, magnesium stearate, ọka starch na lactose monohydrate.

Ere ọgwụ na efere, iri iberibe. Ngwugwu nwere ike si otu ise blisters.

The mbadamba nwere a na-acha ọcha na agba na a okirikiri udi, convex na otu akụkụ.

The ọgwụ ga-echekwara na a gbara ọchịchịrị, akọrọ ebe nke iru nke ụmụ. The okpomọkụ ekwesịghị gafere iri-na-ise degrees. Adị ndụ - maka ise na ụbọchị nke rụpụta. The ọgwụ nwere ike zụta ọ bụla ahịa ọgwụ enweghị a ọgwụ. Ma echefula na onwe pụrụ iduga-ezighị ezi pụta.

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