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Ọgwụ "Tamsulosin": ntuziaka maka ojiji, price, reviews na analogues

"Tamsulosin" antidizuricescoe bụ ọgwụ edinam na-eji dị ka a symptomatic urinary modulator usoro na urological ọrịa ndị cell-ajọ prostate etuto ahụ agwa. The mmeghachi omume usoro a na kwupụtara a jiri nwayọọ nwayọọ na ọnụ na osisi ike na-eji ire ụtọ muscle nke prostate, nakwa dị ka ntụrụndụ nke eriri afo n'olu. Ke adianade do, e nwere a nhọrọ igbochi urethral Alfa 1a-adrenretseptorov, dapụtara na minimization nke mmetụta hụrụ ihe mgbochi - a eke N'ihi ya nke mmepe nke adenomas.

Pharmacological atụmatụ nke "Tamsulosin"

Absorption nke ọgwụ nọ n'ọrụ Efrata na eriri afọ tract nwere ike ịbụ ruo 100%. Experimentally enen na absorption na-ụba mgbe ewere capsules ozugbo a nri. Ogo assimilation proportional ka oge gafeworonụ kemgbe oriri nke ọgwụ (i.e., e nwere a linear kinetics). Ọnụ ọgụgụ kasị elu ịta nke reactants na na plasma bụ imezu mgbe awa isii (otu dose 400 mg). Otú ọ dị, oge a nwere ike ịdị iche dabere na afọ nke ọrịa.

Ọ na-ahụ kwuru na n'ikuku na N'ezie nke ụbọchị ise, ịta nke mmiri na plasma-abawanye site na 60-70%. Tamsulosin hydrochloride zuru ezu nwayọọ nwayọọ na-abanye na metabolic Filiks: uptake esonyere guzobe ufọk ufene metabolites nke nwere nnukwu selectivity maka Alfa 1a-adrenoceptor.

egosi

Ọgwụ "Tamsulosin" ntụziaka ntuziaka classifies dị ka ihe gị n'ụlọnga maka ọgwụgwọ nke benign prostatic hyperplasia, oké symptomatic (adenoma, dysuria, na ndị ọzọ ala Genital tract ọrịa).

Ebe ọ bụ na-adakarị ọmụmụ ekpugheghi ọ bụla dị oké egwu Jeremaya mere, nke ọzọ bekee nke kwuru na-emepụta ọgwụ otu, mgbe ahụ, e nwere dịghị ihe mgbochi na ngwa nke "tamsulosin" dị ka ihe inyeaka mkpali ọgwụ igbochi nhọrọ Alfa-1a adrenergic ihe nnabata.

Na-atụ aro usoro onunu ogwu na usoro nke ochichi

The enweghị hypotensive mmetụta - a mara mma nke ọgwụ "Tamsulosin". Ntuziaka maka ojiji na-ekwu na ọ dị mkpa ka dose nhọrọ naanị bụghị - zuru ezu ọnụ ndinọ 400 micrograms nke ọgwụ mgbe nri ụtụtụ (2 capsules / mbadamba-erikpu 200 mg ọ bụla, ma ọ bụ 1 Capsule / mbadamba-erikpu 400 mg). Ọzọkwa, a kwa ụbọchị ọnụego dịghị mkpa ka e gbazie, ọbụna ma ọ bụrụ na onye ọrịa na-hụrụ obere deviations na akụrụ ma ọ bụ imeju. O sina dị, na mmalite nke ọgwụgwọ N'ezie ga-kpọkwasịwo ihe kpọmkwem nchoputa iji ewepu-ekwe omume nke prostate cancer. Ọzọkwa na niile n'oge ọgwụgwọ amanyere bụ iwu rectal nyochaa.

Capsules na mbadamba "tamsulosin" na-ekwesịghị na-ata - mebiri nke envelopu nwere ike imetụta ntọhapụ ọnụego nke nọ n'ọrụ reagents. Ozugbo na-ewere ọgwụ na-atụ aro na-aṅụ mmiri. Ọ na-machibidoro iji "Tamsulosin" na supine ọnọdụ.

Ẹdude na-agaghị emeli na contraindications

Ọgwụ "Tamsulosin", ego nke nke, dabere na emeputa na nkwakọ formats, àmà 400-1700 rubles, e mere nanị maka ndị ikom. Ya mere, nnyocha na ya mmetụta na nwa ebu n'afọ na-adịghị na e duziri n'oge ime. naanị ọgwụ a na-nyere maka mbadamba data, ya bụ, nchoputa nke "benign prostatic hyperplasia" kwesịrị itinye na nnyocha (na a amanyere bụ iwu tupu ule maka cancer).

N'etiti megide - hypersensitivity na "Tamsulosin" ọgwụ (User ngwa nwere a zuru ezu ndepụta niile inyeaka reagents). Ọ bụ ekwesighi iji nke kwuru gị n'ụlọnga maka orthostatic hypotension na-adịghị ala ala ọrịa imeju ma ọ bụ akụrụ (dị otú ahụ ikpe, ndị dibịa ga na-eme atụmatụ nwere uru nke eji "tamsulosin" na-ekpebi ókè nke na o kwere omume na-ezighị ezi mmetụta nke a ọgwụgwọ N'ezie).

Na mgbe nile n'ikuku ime ìhè dizziness, mgbe ụfọdụ, dochie semiconscious ala. Ụgbọala na-arụ ọrụ, onye ọkachamara ọrụ abuana a iyi egwu nke ọjọọ, ga-edebe oké ịkpachara anya na ojiji nke umi.

mmetụta

Dị ka ọ bụla ọzọ ọgwụ, e nwere mmetụta na ọgwụ "Tamsulosin" (price nke ndị ahụ ike dị elu, nfụkasị Jeremaya na-adị obere, nke mere na oghom Jeremaya-ewere dị ka a dị ịrịba ama enweghị ọ dịghị mkpa).

Ke ukem na-agwọ ọrịa mmetụta nwere ike iri ebe:

  • isi ọwụwa;
  • iyatesịt nke anụ;
  • oge nke afọ ọsịsa;
  • gbasara obi arrhythmias;
  • pelvic mgbu.

"Tamsulosin" Mgbe ụfọdụ, analogues nke ndị a dị ọtụtụ ebe na ahịa, na-eme ehighị ụra nke ọma ọrịa ma ọ bụ, ọzọ, oké ụra. Na obere okwu - a nwa oge mebiri nke oche na-agwụ ike nke potency.

Ovadozu, ya ngosipụta na neutralization

Mgbaàmà nke ovadozu, nke ghọọ a N'ihi ya nke ọgwụ bụ "Tamsulosin" (ntuziaka maka ojiji na aka nke a), ọ nwere ike na-akpọ nnukwu hypotension. Na ọ bụ ezie na likelihood nke a dịruru ná njọ bụ nnọọ ala, na algọridim aka o mere:

  • ozugbo inye onye ọrịa a kehoraizin ọnọdụ;
  • ma ọ bụrụ na ọ dị mkpa, mepụta a mgbagwoju nke jikoro iji na normalisation nke obi usoro nke ahu;
  • iji nyochaa ọrụ nke akụrụ (njikọ ngwa nke wuru ọbara ọcha impractical n'ihi na-arụsi ọrụ ike mgwa ihe n'ụzọ zuru okè metụtara na plasma protein ogige);
  • ime ka vomiting na a ndidi iji kwụsị n'ihu absorption nke reactants (bụkwa eziokwu gastric lavage na yiri iji ihe laxatives);
  • na-anọghị nke Ọnọdụ nke mma itinye ọgwụ ndị na-akpali ọbara ekesa.

Drug interactions: ọdịdị nke Jeremaya mere

"Warfarin" na "Diclofenac" qualitatively emetụta mmepụta ọsọ nke ahụ "Tamsulosin" ọgwụ (ọgwụ price bukwanu, ma pụta bụ uru ọ). Otú ọ dị, ruo ogologo oge kwuru banyere nkwonkwo ihe ndị a ọgwụ ọjọọ eme ihe na ụlọ ọgwụ na-adịghị rụrụ, dị ka a na ya pụta, oké ịkpachara anya na-atụ aro. "Atenolol" na "Enalapril" adịghị emekọ kwuru ihe onwunwe, "cimetidine" akwalite ịta "tamsulosin" plasma, na "Furosemide" enye kpamkpam abụghị N'ihi.

The usoro nke ẹsụhọde ọbara mgbali iwe na oriri nke agwọ ọrịa nwere ike enwekwukwa ruru ka concurrent ojiji nke ọzọ Alfa-1a adrenoblokatorovv ma ọ bụ diuretics na ọgwụ na-akụnwụ. Ịrịba Ama mmetụta na pharmacological kinetics nke free fractions "Diazepam" na "chlormadinone" by nkwadebe "Tamsulosin" ntụziaka ntuziaka (price n'elu n'aka -. 500-1400 ete) na-adịghị kọwaa.

Nchekwa na ọnọdụ na adị ndụ

Na nchekwa ọnọdụ nke ọgwụ "Tamsulosin" nduzi na-ekwu na-esonụ:

  • mma okpomọkụ nso - 15-25 degrees Celsius;
  • kacha iru mmiri - 70%.

Mkpa bụ nchekwa ihe na mbụ nkwakọ (n'ebe a na-apụghị iru bụ ụmụ, nke na-ọma-echebe site kpọmkwem ìhè anyanwụ).

Mgbe niile ihe ntụziaka emeputa di na ọgwụgwọ mmetụta "Tamsulosin" agaghị imeda na afọ abụọ kemgbe ya tọhapụ.

Drug analogues "Tamsulosin"

The ndepụta "mmadụ abụọ" na-anọchi anya abụọ iche iche nke ọgwụ ọjọọ. The mbụ gụnyere ọgwụ ọjọọ, nkịtị, nke abụọ - a obere ahia aha.

Public ego:

  • "Omnic" (na mbụ - Omnic), na-emeputa - na Netherlands, ntọhapụ ụdị - mbadamba / capsules 10/30 iberibe kwa mkpọ, price nso - 380-1700 rubles.
  • "Proflosin" (Proflosin), Germany, blisters nke 30 capsules, ọnụ na-eri - 500 rubles.
  • "Sonizin" (Sonizin), Country nke si malite - Romania, a ọkọlọtọ ngwugwu nke 10 ma ọ bụ 30 capsules, nkezi price - 450 rubles.

Ụghalaahịa ndị ọzọ na ahia aha nke ọgwụ "Tamsulosin" (analogs na ndị na-erughị nkịtị ma ọ bụ hapụ forms ugbua e si mmepụta):

  • "Omsulozin" (Omsulosin), India, capsules 0.4 mg (30 PC.) Price ranges si 350 na 550 rubles.
  • "Tamsulosin-Teva" (Tamsulosin-Teva), "Tema-Actavis" ụlọ ọrụ na ngwaahịa, Greece, udi nke mkpo ya na price bụ otu ihe ahụ dị ka na aga na ikpe.
  • "Tamsulosin-ghara" ( "understudy" nyere ntọhapụ akụrụngwa), mmepụta akara biri na Russia, mbadamba 400 mg, ndị na-eri - banyere 300-360 rubles.

"Tamsulosin": reviews nke dọkịta na ndị ọrịa

Medical ọgwụ na a ọgwụ bụ n'ozuzu ịga nke ọma ma na-kwupụtara a nlaghachi azụ okwu pụta ụwa na-abụghị ndị ajọ prostate etuto ahụ.

Mgbe ihe 90 ụbọchị nke mgbaàmà e belata na 2 ugboro, na nke mbụ kwesiri ngosi mgbanwe na-ama hụrụ n'ụlọ 14-21 ụbọchị. N'elu ẹkụre nke mgbaàmà nke index Falls 75% (tụnyere na-amalite na-adọ), nke bụ na-na-anara nke N'ihi.

Mara mma tolerability "Tamsulosin" (ndu price na ọtụtụ nkịtị ọnyà ọgwụ ọjọọ na-e nyere n'elu) na-eme ka ọ dị nnọọ adaba iji mgbe na-ekenye ndị ọrịa na ọgwụgwọ. Otú ọ dị, iji nweta kacha nwere mmetụta nke umi na-ezughi oke, ọ na-atụ aro na concurrent ọgwụ na ụzọ ndị ọzọ na-emepụta ọgwụ na ngwaahịa.

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